Life Science / Inhibitors/Agonists / Apoptosis / Caspase

Cat. No. Name/Description Purity
A622861 Emricasan

98%
A737788 Arnicolide D

97%
A426528 Ac-DEVD-CHO

97%
A230023 Aristolactam I

97%
A239560 Dehydrocorydaline chloride

98%
A834991 Z-VAD-FMK

98%
A390989 5,7-Dihydroxychromone

98%
A100567 VX-765

99%
A149084 Akebia saponin D

98%
A574284 GRI977143

95%
A169042 Azoramide

98%
A131202 PAC-1

98%
A1209725 Boc-Asp(OMe)-fluoromethyl ketone

90%
A724295 2-HBA

98%
A1339274 Procaspase-3/6 activator 1

98+%
A354225 Z-VAD(OMe)-FMK

98%
A505764 5-TAMRA

98%
A301584 Z-DEVD-FMK

98%
A553186 Ossirene

98%
A173783 Taurodeoxycholic acid sodium hydrate

95%

No Data

Name/Description Capase-7 Caspase Caspase-1 Caspase-10 Caspase-2 Caspase-3 Caspase-4 Caspase-5 Caspase-6 Caspase-8 Caspase-9 Other Targets Purity
Ac-DEVD-CHO +++

caspase-7, Ki: 1.6 nM

+++

Caspase-1, Ki: 18 nM

+++

caspase-10, Ki: 12 nM

+

caspase-2, Ki: 1.71 μM

++++

Caspase-3, Ki: 230 pM

++

Caspase-4, Ki: 132 nM

++

caspase-5, Ki: 205 nM

+++

caspase-6, Ki: 31 nM

++++

caspase-8, Ki: 0.92 nM

++

Caspase-9, Ki: 60 nM

99%+
Emricasan 99%+
Z-VAD(OMe)-FMK 99%+
Z-VAD-FMK 99%+
Z-DEVD-FMK 99%+
VX-765 ++++

Caspase-1, Ki: 0.8 nM

++++

Caspase-4, Ki: <0.6 nM

99%+
Q-VD-OPh 97%
Z-IETD-FMK 99%+
1. Hovering the mouse over the "+" can display the specific value of the relevant IC50. The more "+", the stronger the inhibitory effect. 2. "✔" Indicates that the compound has inhibitory effects on the corresponding subtypes, but there is currently no relevant data on the intensity of inhibition.