Life Science / Inhibitors/Agonists / Metabolic Enzyme / PDE

Cat. No. Name/Description Purity
A111758 N-Methylbenzamide

97%
A304814 MY-5445

98%
A273394 Ayanin

98%
A982733 (E/Z)-Ensifentrine

98%
A505170 Zardaverine

98%
A656644 TBA-7371

98%
A570430 5,7-Diacetoxy-8-methoxyflavone

98%
A144390 3,?5,?6,?7,?8,?3',?4'-?Heptemthoxyflavone

98%
A217533 Kushenol A

98%
A860292 3-O-Methylquercetin

98%
A541549 GSK256066

98+%
A124931 Yonkenafil

95%
A1176934 Osoresnontrine

99+%
A459882 IBMX

98%
A1500036 (+)-Medioresinol Di-O-β-D-glucopyranoside

98%
A110103 Amrinone

99%
A147960 Tadalafil

98%
A613618 Oglemilast

98%
A1537879 FEN1-IN-SC13

95%
A218047 Milrinone

98%

No Data

Name/Description PDE PDE1 PDE10A PDE2 PDE3 PDE4 PDE5 PDE6 Other Targets Purity
Deltarasin +++

PDEδ , Kd: 38 nM

99+%
7-(2,3-Dihydroxypropyl)theophylline 98%
Anagrelide HCl 99%+
Irsogladine mAChR,AChR 98%
PF-8380 +++

Autotaxin, IC50: 2.8 nM

99%+
Dipyridamole 98%
Balipodect ++++

PDE10A, IC50: 0.3 nM

99%+
PF-2545920 ++++

PDE10A, IC50: 0.37 nM

97%
Luteolin +

PDE1, Ki: 15.0 μM

++

PDE2, Ki: 6.4 μM

+

PDE3, Ki: 13.9 μM

+

PDE4, Ki: 11.1 μM

+

PDE5, Ki: 9.5 μM

98%
Milrinone ++

PDE2, IC50: 5.2 μM

++

PDE3, IC50: 2.1 μM

ATPase 98%
Pimobendan ++

PDE3, IC50: 0.32 μM

98%
Cilostazol ++

PDE3, IC50: 0.2 μM

98%
(S)-(+)-Rolipram ++

PDE4, IC50: 0.75 μM

98%
Apremilast +++

PDE4, IC50: 74 nM

98%
GSK256066 ++++

PDE4B, IC50: 3.2 pM

99%+
Roflumilast ++++

PDE4A4, IC50: 4.3 nM

PDE4A1, IC50: 0.7 nM

99%
Rolipram +++

PDE4B, IC50: 130 nM

99%+
Cilomilast +++

HPDE4, IC50: 120 nM

LPDE4, IC50: 100 nM

98+%
Avanafil ++++

PDE5, IC50: 1 nM

98%
Vardenafil HCl Trihydrate ++++

PDE5, IC50: 0.7 nM

98%
Tadalafil ++++

PDE5, IC50: 1.8 nM

98%
Icariin ++

PDE5, IC50: 0.432 μM

98%
1. Hovering the mouse over the "+" can display the specific value of the relevant IC50. The more "+", the stronger the inhibitory effect. 2. "✔" Indicates that the compound has inhibitory effects on the corresponding subtypes, but there is currently no relevant data on the intensity of inhibition.