Life Science / Inhibitors/Agonists / / ROCK

Cat. No. Name/Description Purity
A225129 Narciclasine

98%
A112358 Y-27632

98%
A255643 Belumosudil

99%
A168750 BAY-549

98%
A266066 GSK269962A

98%
A1165861 CMPD101

98%
A1598869 ROCK1-IN-1

95%
A105790 GSK269962A HCl

98%
A101744 Y-27632 dihydrochloride

99%
A100468 ZINC00881524

98%
A204681 Y-33075 2HCl

98+%
A1213276 CCG-222740

98+%
A1806913 CAY10746

98%
A193859 Fasudil HCl

98%
A130094 Ripasudil

98%
A919821 ROCK2-IN-2

98%
A1229459 ROCK-IN-5

98%
A1263609 Netarsudil Mesylate

98%
A244270 Hydroxyfasudil

98%
A303159 SAR407899

98+%

No Data

Name/Description ROCK ROCK1 ROCK2 Other Targets Purity
Thiazovivin +

ROCK, IC50: ~0.5 μM

98+%
Netarsudil hydrochloride ++++

ROCK, Ki: 2 nM

99%+
Y-33075 2HCl ++++

ROCK, IC50: 3.6 nM

99%+
ROCK1-IN-1 ++

ROCK, Ki: 17nM

95%
GSK429286A +++

ROCK1, IC50: 14 nM

++

ROCK2, IC50: 63 nM

99%+
Ripasudil ++

ROCK1, IC50: 51 nM

++

ROCK2, IC50: 19 nM

99%+
Y-27632 dihydrochloride ++

ROCK1, Ki: 140 nM

+

ROCK2, Ki: 300 nM

99%+
Chroman 1 ++++

ROCK1, IC50: 52 pM

++++

ROCK2, IC50: 1 pM

99%
BAY-549 ++++

ROCK1, IC50: 0.6 nM

++++

ROCK2, IC50: 1.1 nM

98%+
RKI-1447 +++

ROCK1, IC50: 14.5 nM

+++

ROCK2, IC50: 6.2 nM

99%+
Hydroxyfasudil HCl +

ROCK1, IC50: 0.73 μM

+

ROCK2, IC50: 0.72 μM

PKA 99%+
GSK269962A HCl ++++

ROCK1, IC50: 1.6 nM

+++

ROCK2, IC50: 4 nM

99%+
Belumosudil ++

ROCK2, IC50: 60 nM

ROCK2, Ki: 41 nM

99%+
Fasudil HCl +

ROCK2, Ki: 330 nM

Rho,PKG 98%
H-1152 2HCl +++

ROCK2, IC50: 0.0120 μM

PKG 99%
1. Hovering the mouse over the "+" can display the specific value of the relevant IC50. The more "+", the stronger the inhibitory effect. 2. "✔" Indicates that the compound has inhibitory effects on the corresponding subtypes, but there is currently no relevant data on the intensity of inhibition.