Cat. No. | Name/Description | Purity |
---|---|---|
A225129 | Narciclasine | 98% |
A112358 | Y-27632 | 98% |
A255643 | Belumosudil | 99% |
A168750 | BAY-549 | 98% |
A266066 | GSK269962A | 98% |
A1165861 | CMPD101 | 98% |
A1598869 | ROCK1-IN-1 | 95% |
A105790 | GSK269962A HCl | 98% |
A101744 | Y-27632 dihydrochloride | 99% |
A100468 | ZINC00881524 | 98% |
A204681 | Y-33075 2HCl | 98+% |
A1213276 | CCG-222740 | 98+% |
A1806913 | CAY10746 | 98% |
A193859 | Fasudil HCl | 98% |
A130094 | Ripasudil | 98% |
A919821 | ROCK2-IN-2 | 98% |
A1229459 | ROCK-IN-5 | 98% |
A1263609 | Netarsudil Mesylate | 98% |
A244270 | Hydroxyfasudil | 98% |
A303159 | SAR407899 | 98+% |
Name/Description | ROCK ↓ ↑ | ROCK1 ↓ ↑ | ROCK2 ↓ ↑ | Other Targets | Purity | ||||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Thiazovivin |
+
ROCK, IC50: ~0.5 μM |
98+% | |||||||||||||||||
Netarsudil hydrochloride |
++++
ROCK, Ki: 2 nM |
99%+ | |||||||||||||||||
Y-33075 2HCl |
++++
ROCK, IC50: 3.6 nM |
99%+ | |||||||||||||||||
ROCK1-IN-1 |
++
ROCK, Ki: 17nM |
95% | |||||||||||||||||
GSK429286A |
+++
ROCK1, IC50: 14 nM |
++
ROCK2, IC50: 63 nM |
99%+ | ||||||||||||||||
Ripasudil |
++
ROCK1, IC50: 51 nM |
++
ROCK2, IC50: 19 nM |
99%+ | ||||||||||||||||
Y-27632 dihydrochloride |
++
ROCK1, Ki: 140 nM |
+
ROCK2, Ki: 300 nM |
99%+ | ||||||||||||||||
Chroman 1 |
++++
ROCK1, IC50: 52 pM |
++++
ROCK2, IC50: 1 pM |
99% | ||||||||||||||||
BAY-549 |
++++
ROCK1, IC50: 0.6 nM |
++++
ROCK2, IC50: 1.1 nM |
98%+ | ||||||||||||||||
RKI-1447 |
+++
ROCK1, IC50: 14.5 nM |
+++
ROCK2, IC50: 6.2 nM |
99%+ | ||||||||||||||||
Hydroxyfasudil HCl |
+
ROCK1, IC50: 0.73 μM |
+
ROCK2, IC50: 0.72 μM |
PKA | 99%+ | |||||||||||||||
GSK269962A HCl |
++++
ROCK1, IC50: 1.6 nM |
+++
ROCK2, IC50: 4 nM |
99%+ | ||||||||||||||||
Belumosudil |
++
ROCK2, IC50: 60 nM ROCK2, Ki: 41 nM |
99%+ | |||||||||||||||||
Fasudil HCl |
+
ROCK2, Ki: 330 nM |
Rho,PKG | 98% | ||||||||||||||||
H-1152 2HCl |
+++
ROCK2, IC50: 0.0120 μM |
PKG | 99% | ||||||||||||||||
1. Hovering the mouse over the "+" can display the specific value of the relevant IC50. The more "+", the stronger the inhibitory effect. 2. "✔" Indicates that the compound has inhibitory effects on the corresponding subtypes, but there is currently no relevant data on the intensity of inhibition. |