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Chemical Structure| 2543545-44-2 Chemical Structure| 2543545-44-2

Structure of LT052
CAS No.: 2543545-44-2

Chemical Structure| 2543545-44-2

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LT052 is a highly selective BET BD1 inhibitor with an IC50 of 87.7 nM, exhibiting nanomolar-level inhibition of BRD4 BD1, with 138 times selectivity over BRD4 BD2 (IC50 = 12.130 μM). LT052 exhibits anti-inflammatory activity and can be used for acute gouty arthritis research.

Synonyms: LT052

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Product Details of LT052

CAS No. :2543545-44-2
Formula : C22H19N5O4S
M.W : 449.48
SMILES Code : O=S(C1=CC=CC=C1OC)(NC2=C3N=C(N4C=C(C)N=C4)C=C5C3=C(N(C)C5=O)C=C2)=O
Synonyms :
LT052

Safety of LT052

GHS Pictogram:
Signal Word:Warning
Hazard Statements:H302-H315-H319
Precautionary Statements:P501-P270-P264-P280-P302+P352-P337+P313-P305+P351+P338-P362+P364-P332+P313-P301+P312+P330

Related Pathways of LT052

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Preparing Stock Solutions 1mg 5mg 10mg

1 mM

5 mM

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2.22mL

0.44mL

0.22mL

11.12mL

2.22mL

1.11mL

22.25mL

4.45mL

2.22mL

 

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