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Chemical Structure| 1256937-27-5 Chemical Structure| 1256937-27-5

Structure of Evolocumab
CAS No.: 1256937-27-5

Chemical Structure| 1256937-27-5

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Evolocumab is a humanized IgG2 monoclonal antibody that prevents PCSK9 from binding to LDL receptors. Evolocumab has potential for research on hypercholesterolemia.

Synonyms: AMG 145

4.5 *For Research Use Only !

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Product Details of Evolocumab

CAS No. :1256937-27-5
M.W : 141.8 kDa
SMILES Code : NONE
Synonyms :
AMG 145

Safety of Evolocumab

GHS Pictogram:
Signal Word:Warning
Hazard Statements:H302-H315-H319
Precautionary Statements:P501-P270-P264-P280-P302+P352-P337+P313-P305+P351+P338-P362+P364-P332+P313-P301+P312+P330

Isoform Comparison

Biological Activity

Clinical Trial:

NCT Number Conditions Phases Recruitment Completion Date Locations
NCT05697185 Ischemic Stroke, Acute PHASE4 UNKNOWN 2024-12-01 -
NCT03791593 Heart Failure With Reduced Eje... More >>ction Fraction Less << PHASE2 COMPLETED 2022-07-20 Hospital Universitari Germans ... More >>Trias i Pujol, Badalona, Barcelona, 08916, Spain|Hospital Universitario Virgen del Rocío, Sevilla, 41013, Spain|Hospital Clínico de Valencia, Valencia, 46010, Spain Less <<
NCT05152888 Stable Coronary Disease PHASE4 RECRUITING 2025-12-31 Brigham and Women's Hospital, ... More >>Boston, Massachusetts, 02115, United States Less <<
NCT02948777 Type 2 Diabetes Mellitus PHASE4 COMPLETED 2025-06-18 Helsinki University Hospital, ... More >>Biomedicum 2U, Helsinki, Finland Less <<
NCT05579418 STEMI|Dyslipidemias PHASE4 UNKNOWN 2024-10-30 -
NCT03500302 Human Immunodeficiency Virus|C... More >>oronary Artery Disease Less << PHASE2 COMPLETED 2019-11-30 Johns Hopkins University, Balt... More >>imore, Maryland, 21205, United States Less <<
NCT03080935 Dyslipidemia PHASE3 TERMINATED 2022-03-04 Algemeen Stedelijk Ziekenhuis ... More >>Aalst, Aalst, 9300, Belgium|Onze Lieve Vrouw Ziekenhuis Aalst, Aalst, 9300, Belgium|Ziekenhuis Netwerk Antwerpen Middelheim, Antwerpen, 2020, Belgium|Ziekenhuis Netwerk Antwerpen Stuivenberg, Antwerpen, 2060, Belgium|Imelda Ziekenhuis vzw, Bonheiden, 2820, Belgium|Centre Hospitalier Universitaire Brugmann, Brussels, 1020, Belgium|Cliniques universitaires de Bruxelles Hopital Erasme, Brussels, 1070, Belgium|Universite Catholique de Louvain Cliniques Universitaires Saint Luc, Bruxelles, 1200, Belgium|Algemeen Ziekenhuis Sint Lucas, Gent, 9000, Belgium|Universitair Ziekenhuis Gent, Gent, 9000, Belgium|Medif sprl, Gozee, 6534, Belgium|Centre Hospitalier Universitaire de Tivoli, La Louvi?¨re, 7100, Belgium|Centres Hospitaliers Jolimont - Hopital de Jolimont, La Louvi?¨re, 7100, Belgium|Centre Hospitalier Universitaire de Liege - Sart Tilman, Liege, 4000, Belgium|Centre Hospitalier Regional de la Citadelle, Li?¨ge, 4000, Belgium|Algemeen Ziekenhuis Turnhout, Turnhout, 2300, Belgium|Aalborg Hospital, Aalborg, 9000, Denmark|Center for Clinical and Basic Research Aalborg, Aalborg, 9000, Denmark|Aarhus Universitetshospital, Aarhus N, 8200, Denmark|Centre for Clinical and Basic Research Ballerup, Ballerup, 2750, Denmark|Sydvestjysk Sygehus, Esbjerg, 6700, Denmark|Frederiksberg/Bispebjerg Hospitaler, Frederiksberg, 2000, Denmark|Glostrup Hospital, Glostrup, 2600, Denmark|Hvidovre Hospital, Hvidovre, 2650, Denmark|Amager Hospital, Kobenhavn S, 2300, Denmark|Odense Universitetssygehus, Odense, 5000, Denmark|Sjaellands Universitetshospital, Roskilde, Roskilde, 4000, Denmark|Svendborg Sygehus, Svendborg, 5700, Denmark|Center for Clinical and Basic Research Vejle, Vejle, 7100, Denmark|Regionshospitalet Viborg, Viborg, 8800, Denmark|Centre Hospitalier Regional Universitaire de Besancon, Hopital Jean Minjoz, Besancon cedex, 25030, France|Centre Hospitalier R??gional Universitaire de Tours - H?′pital Trousseau, Chambray les Tours, 37170, France|Hopital Louis Pasteur, Le Coudray, 28630, France|Centre Hospitalier Regional Universitaire de Montpellier - Hopital Arnaud de Villeneuve, Montpellier cedex 05, 34295, France|Centre Hospitalier Universitaire de Nantes - Hopital Guillaume et Rene Laennec, Nantes Cedex 1, 44093, France|Nouvelles Cliniques Nantaises, Nantes Cedex 2, 44202, France|Centre Hospitalier Universitaire de Nice - Hopital Pasteur, Nice, 06000, France|Hopital Lariboisiere, Paris, 75010, France|Hopital Pitie-Salpetriere, Paris, 75013, France|Centre Hospitalier de Pau - Hopital Francois Mitterrand, Pau, 64000, France|Centre Hospitalier Universitaire de Reims - Hopital Robert Debre, Reims, 51100, France|Centre Hospitalier Universitaire de Toulouse - Hopital Rangueil, Toulouse Cedex 9, 31059, France|Centre Hospitalier Intercommunal Haute Saone, Vesoul, 70014, France|Universitaets-Herzzentrum Freiburg - Bad Krozingen, Bad Krozingen, 79189, Germany|Klinische Forschung Berlin GbR, Berlin, 10787, Germany|Vivantes Klinikum Neuk??lln, Berlin, 12351, Germany|Deutsches Rotes Kreuz Kliniken Berlin K??penick, Berlin, 12559, Germany|Deutsches Herzzentrum Berlin, Berlin, 13353, Germany|Sankt-Johannes-Hospital, Dortmund, 44137, Germany|Gesellschaft fur Wissens und Technologietransfer der Technischen Uni Dresden, Dresden, 01307, Germany|Ambulantes Herzzentrum Kassel, Kassel, 34121, Germany|Universit?¤tsklinikum K??ln, K??ln, 50937, Germany|Otto von Guericke Universit?¤t Magdeburg, Magdeburg, 39120, Germany|Johannes Gutenberg Universit?¤t Mainz, Mainz, 55131, Germany|Herz-Gef?¤??-Zentrum Nymphenburg am Klinikum Dritter Orden, M??nchen, 80333, Germany|Deutsches Herzzentrum M??nchen des Freistaates Bayern, M??nchen, 80636, Germany|Robert Bosch Krankenhaus, Stuttgart, 70376, Germany|Universit?¤tsklinikum Ulm, Ulm, 89081, Germany|Forschungszentrum Ruhr, Witten, 58455, Germany|Helios Universit?¤tsklinikum Wuppertal, Wuppertal, 42117, Germany|Azienda Socio Sanitaria Territoriale Papa Giovanni XXIII, Bergamo, 24127, Italy|Azienda Ospedaliero Universitaria Careggi, Firenze, 50139, Italy|Centro Cardiologico Monzino, Milano, 20138, Italy|Azienda Socio Sanitaria Territoriale Grande Ospedale Metropolitano Niguarda, Milano, 20162, Italy|Azienda Ospedaliera Ospedali Riuniti Villa Sofia Cervello, Palermo, 90146, Italy|Fondazione IRCCS Policlinico San Matteo, Pavia, 27100, Italy|Azienda Ospedaliera di Perugia Ospedale Santa Maria della Misericordia, Perugia, 06129, Italy|Fondazione Toscana Gabriele Monasterio, Stabilimento Ospedaliero di Pisa, Pisa, 56124, Italy|Azienda Ospedaliera Universitaria Senese Policlinico Le Scotte, Siena, 53100, Italy|Hospital Garcia de Orta, EPE, Almada, 2801-951, Portugal|Centro Hospitalar e Universitario de Coimbra EPE, Coimbra, 3000-075, Portugal|Centro Hospitalar Cova da Beira, EPE - Hospital Pero da Covilha, Covilha, 6200-251, Portugal|Hospital Cuf Infante Santo, Lisboa, 1350-352, Portugal|Centro Hospitalar de Lisboa Ocidental, EPE - Hospital Sao Francisco Xavier, Lisboa, 1449-005, Portugal|Centro Hospitalar de Setubal EPE Hospital de Sao Bernardo, Setubal, 2910-446, Portugal|Falu Lasarett, Falun, 791 82, Sweden|Helsingborgs Lasarett, Helsingborg, 252 47, Sweden|L?¤nssjukhuset Ryhov, J??nk??ping, 551 85, Sweden|Sunderby Sjukhus, Lulea, 971 80, Sweden|Skanes Universitetssjukhus, Lund, 221 85, Sweden|Capio Citykliniken, Lund, 222 21, Sweden|Universitetssjukhuset ?-rebro, Orebro, 701 85, Sweden|Ostersunds sjukhus, Ostersund, 831 83, Sweden|Akardo MedSite, Stockholm, 117 27, Sweden|Norrlands Universitetssjukhus, Umea, 901 85, Sweden Less <<
NCT04087915 Dyslipidemia|High Risk Coronar... More >>y Artery Disease Less << UNKNOWN 2021-12-31 Beijing Anzhen Hospital, Capit... More >>al Medical University, Beijing, Beijing, 100029, China Less <<
NCT05418166 Acute Coronary Syndrome UNKNOWN 2022-09-01 the first affiliated hospital ... More >>of Harbin Medical University, Harbin, Heilongjiang, 150000, China Less <<
NCT03247972 Peripheral Arterial Disease TERMINATED 2019-10-01 Inova Fairfax Hospital, Falls ... More >>Church, Virginia, 22042, United States Less <<
NCT03331666 Familial Hypercholesterolemia PHASE4 TERMINATED 2020-02-04 Columbia University Medical Ce... More >>nter, New York, New York, 10032, United States Less <<
NCT03944577 Heart Transplant PHASE2 COMPLETED 2023-03-28 University of Nebraska Medical... More >> Center, Omaha, Nebraska, 68198, United States Less <<
NCT04665830 Kideny Transplant Recipients W... More >>ith High Cardiovascular Risk Score Less << PHASE3 COMPLETED 2020-05-01 OTC, MOH , Kuwait, Kuwait, Kuw... More >>ait, Kuwait Less <<
NCT06140095 Acute Metabolic Effects of Evo... More >>locumab and Atorvastatin Less << EARLY_PHASE1 NOT_YET_RECRUITING 2025-12-25 -
NCT04100434 Acute Coronary Syndrome|Propro... More >>tein Convertase Subtilisin/Kexin Type 9 Inhibitor Less << PHASE4 UNKNOWN 2023-06-01 Tianjin Chest Hospital,, Tianj... More >>in, 300222, China Less <<
NCT06231459 Hypercholesterolemia, Familial PHASE4 COMPLETED 2020-12-31 National Medical Center "20 de... More >> Noviembre", ISSSTE, Mexico City, 03100, Mexico Less <<
NCT04313270 Hypercholesterolemia, Familial RECRUITING 2025-12-01 Matteo Di Minno, Napoli, 80131... More >>, Italy Less <<
NCT04937413 Malignant Glioma|Glioblastoma EARLY_PHASE1 COMPLETED 2023-10-12 Duke University Medical Center... More >>, Durham, North Carolina, 27710, United States Less <<
NCT04539223 Carotid Artery Stenosis|Asympt... More >>omatic Carotid Artery Stenosis Less << PHASE4 UNKNOWN 2025-05-22 North York Diagnostic and Card... More >>iac Centre, North York, Ontario, M6B 3H7, Canada|East Toronto Vascular Clinic, Toronto, Ontario, M4L3Y3, Canada|St. Michael's Hospital, Toronto, Ontario, Canada Less <<
 

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