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Chemical Structure| 1644670-37-0 Chemical Structure| 1644670-37-0

Structure of Iptacopan
CAS No.: 1644670-37-0

Chemical Structure| 1644670-37-0

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Iptacopan is a pioneering, efficient, orally active factor B inhibitor with an IC50 of 10 nM and a KD of 7.9 nM. It directly and reversibly binds to factor B, targeting the root cause of C3 glomerulopathy, demonstrating substantial therapeutic potential for such diseases.

Synonyms: LNP023

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Product Details of Iptacopan

CAS No. :1644670-37-0
Formula : C25H30N2O4
M.W : 422.52
SMILES Code : [H][C@@]1(C2=CC=C(C(O)=O)C=C2)C[C@@H](OCC)CCN1CC3=C4C=CNC4=C(C)C=C3OC
Synonyms :
LNP023
MDL No. :MFCD32174282

Safety of Iptacopan

GHS Pictogram:
Signal Word:Warning
Hazard Statements:H315-H319
Precautionary Statements:P264-P280-P302+P352-P337+P313-P305+P351+P338-P362+P364-P332+P313

Isoform Comparison

Biological Activity

Clinical Trial:

NCT Number Conditions Phases Recruitment Completion Date Locations
NCT05222412 C3 Glomerulopathy (C3G)|Paroxy... More >>smal Nocturnal Hemoglobinuria (PNH) Less << AVAILABLE - -
NCT03955445 C3 Glomerulopathy|Idiopathic I... More >>mmune-complex-membranoproliferative Glomerulonephritis Less << PHASE3 RECRUITING 2033-04-20 Georgia Nephrology Research In... More >>st, Lawrenceville, Georgia, 30046, United States|University of Iowa Health Care, Iowa City, Iowa, 52242-1091, United States|Col Uni Med Center New York Presby, New York, New York, 10032, United States|Novartis Investigative Site, Buenos Aires, W3400ABH, Argentina|Novartis Investigative Site, Sao Paulo, SP, 04038-002, Brazil|Novartis Investigative Site, Toronto, Ontario, M5G 2C4, Canada|Novartis Investigative Site, Beijing, 100034, China|Novartis Investigative Site, Shanghai, 200040, China|Novartis Investigative Site, Praha, 12808, Czechia|Novartis Investigative Site, Montpellier Cedex 5, 34295, France|Novartis Investigative Site, Paris 15, 75015, France|Novartis Investigative Site, Paris, 75015, France|Novartis Investigative Site, Erlangen, 91054, Germany|Novartis Investigative Site, Essen, 45147, Germany|Novartis Investigative Site, Hamburg, 20246, Germany|Novartis Investigative Site, Heraklion Crete, 71110, Greece|Novartis Investigative Site, Petach Tikva, 49202, Israel|Novartis Investigative Site, Petach Tikva, 4941492, Israel|Novartis Investigative Site, Ranica, BG, 24020, Italy|Novartis Investigative Site, Roma, RM, 00165, Italy|Novartis Investigative Site, Nagoya, Aichi, 466 8560, Japan|Novartis Investigative Site, Asahikawa, Hokkaido, 078 8510, Japan|Novartis Investigative Site, Sapporo, Hokkaido, 060-8543, Japan|Novartis Investigative Site, Takatsuki, Osaka, 569 1192, Japan|Novartis Investigative Site, Niigata, 951 8520, Japan|Novartis Investigative Site, Leiden, Zuid Holland, 2333 ZA, Netherlands|Novartis Investigative Site, Sevilla, Andalucia, 41009, Spain|Novartis Investigative Site, Barcelona, Catalunya, 08035, Spain|Novartis Investigative Site, Pamplona, Navarra, 31008, Spain|Novartis Investigative Site, Madrid, 28040, Spain|Novartis Investigative Site, Madrid, 28041, Spain|Novartis Investigative Site, Bern, 3010, Switzerland|Novartis Investigative Site, Ankara, 06500, Turkey|Novartis Investigative Site, Talas Kayseri, 38039, Turkey|Novartis Investigative Site, London, W12 0HS, United Kingdom|Novartis Investigative Site, Newcastle upon Tyne, NE7 7DN, United Kingdom Less <<
NCT04557462 Primary IgA Nephropathy PHASE3 RECRUITING 2032-10-28 AZ Kidney Dise and Hypertensio... More >>n Ctr, Glendale, Arizona, 85306, United States|Kaiser Permanente, San Diego, California, 92111, United States|North America Research Institute, San Dimas, California, 91773, United States|University of Colorado Anschutz, Aurora, Colorado, 80045, United States|Nephrology Associates PA, Newark, Delaware, 19713, United States|CaRe Research, Chubbuck, Idaho, 83202, United States|Brigham and Womens Hosp Harvard Med School, Boston, Massachusetts, 02115, United States|Clinical Research Consultants LLC, Kansas City, Missouri, 64111, United States|DaVita Clinical Research, Las Vegas, Nevada, 89146, United States|Prolato Clinical Research Center, Houston, Texas, 77054, United States|Novartis Investigative Site, Ciudad Autonoma de Buenos Aire, 1426, Argentina|Novartis Investigative Site, Cordoba, X5016KET, Argentina|Novartis Investigative Site, Santa Fe, S3000EPV, Argentina|Novartis Investigative Site, Woolloongabba, Queensland, 4102, Australia|Novartis Investigative Site, Adelaide, South Australia, 5000, Australia|Novartis Investigative Site, Parkville, Victoria, 3065, Australia|Novartis Investigative Site, Edegem, 2650, Belgium|Novartis Investigative Site, Leuven, 3000, Belgium|Novartis Investigative Site, Roeselare, 8800, Belgium|Novartis Investigative Site, Curitiba, PR, 80440-020, Brazil|Novartis Investigative Site, Porto Alegre, RS, 90020-090, Brazil|Novartis Investigative Site, Sao Paulo, SP, 04038-002, Brazil|Novartis Investigative Site, Sao Paulo, SP, 05403 000, Brazil|Novartis Investigative Site, Sao Jose do Rio Preto, 15090 000, Brazil|Novartis Investigative Site, Oshawa, Ontario, L1G 2B9, Canada|Novartis Investigative Site, Guangzhou, Guangdong, 510080, China|Novartis Investigative Site, Changchun, Jilin, 130041, China|Novartis Investigative Site, Yinchuan, Ningxia, 100039, China|Novartis Investigative Site, Taiyuan, Shanxi, 030001, China|Novartis Investigative Site, Wenzhou, Zhejiang, 325000, China|Novartis Investigative Site, Beijing, 100029, China|Novartis Investigative Site, Beijing, 100034, China|Novartis Investigative Site, Guang Zhou, 510080, China|Novartis Investigative Site, Qingdao, 266000, China|Novartis Investigative Site, Shanghai, 200025, China|Novartis Investigative Site, Shanghai, 200040, China|Novartis Investigative Site, Shanxi, 710063, China|Novartis Investigative Site, Shenzhen, 518036, China|Novartis Investigative Site, Medellin, Antioquia, 050001, Colombia|Novartis Investigative Site, Praha, 12808, Czechia|Novartis Investigative Site, Aalborg, 9000, Denmark|Novartis Investigative Site, Arhus N, DK-8200, Denmark|Novartis Investigative Site, Copenhagen, DK-2100, Denmark|Novartis Investigative Site, Odense C, 5000, Denmark|Novartis Investigative Site, Marseille, 13385, France|Novartis Investigative Site, Paris, 75015, France|Novartis Investigative Site, Aachen, 52074, Germany|Novartis Investigative Site, Berlin, 13353, Germany|Novartis Investigative Site, Freiburg, 79106, Germany|Novartis Investigative Site, Heidelberg, 69120, Germany|Novartis Investigative Site, Magdeburg, 39120, Germany|Novartis Investigative Site, Mainz, 55131, Germany|Novartis Investigative Site, Tuebingen, 72076, Germany|Novartis Investigative Site, Ulm, 89081, Germany|Novartis Investigative Site, Pokfulam, Hong Kong|Novartis Investigative Site, Debrecen, 4032, Hungary|Novartis Investigative Site, Bangalore, Karnataka, 560004, India|Novartis Investigative Site, New Delhi, 110029, India|Novartis Investigative Site, Ashkelon, 78278, Israel|Novartis Investigative Site, Jerusalem, 9112001, Israel|Novartis Investigative Site, Petach Tikva, 4941492, Israel|Novartis Investigative Site, Napoli, 80131, Italy|Novartis Investigative Site, Kasugai, Aichi, 486-8510, Japan|Novartis Investigative Site, Toyoake city, Aichi, 470 1192, Japan|Novartis Investigative Site, Toyota, Aichi, 471-8513, Japan|Novartis Investigative Site, Sapporo-city, Hokkaido, 006-8555, Japan|Novartis Investigative Site, Sapporo, Hokkaido, 060-8604, Japan|Novartis Investigative Site, Kawasaki, Kanagawa, 213-8587, Japan|Novartis Investigative Site, Yokohama-city, Kanagawa, 236-0004, Japan|Novartis Investigative Site, Yokohama, Kanagawa, 224-8503, Japan|Novartis Investigative Site, Sendai, Miyagi, 981-3205, Japan|Novartis Investigative Site, Matsumoto, Nagano, 390-8621, Japan|Novartis Investigative Site, Okayama-city, Okayama, 700-8558, Japan|Novartis Investigative Site, Omihachiman, Shiga, 523-0082, Japan|Novartis Investigative Site, Chiba, 260-8712, Japan|Novartis Investigative Site, Kyoto, 605-0981, Japan|Novartis Investigative Site, Osaka, 530-0012, Japan|Novartis Investigative Site, Osaka, 530-8480, Japan|Novartis Investigative Site, Osaka, 534-0021, Japan|Novartis Investigative Site, Cheongju si, Chungcheongbuk Do, 28644, Korea, Republic of|Novartis Investigative Site, Seoul, Korea, 03312, Korea, Republic of|Novartis Investigative Site, Seoul, Seocho Gu, 06591, Korea, Republic of|Novartis Investigative Site, Busan, 47392, Korea, Republic of|Novartis Investigative Site, Seoul, 02841, Korea, Republic of|Novartis Investigative Site, Seoul, 03080, Korea, Republic of|Novartis Investigative Site, Seoul, 03722, Korea, Republic of|Novartis Investigative Site, Seoul, 06973, Korea, Republic of|Novartis Investigative Site, Seoul, 134 727, Korea, Republic of|Novartis Investigative Site, Taegu, 41944, Korea, Republic of|Novartis Investigative Site, Kuala Lumpur, Wilayah Persekutuan, 50586, Malaysia|Novartis Investigative Site, Kuala Lumpur, 59100, Malaysia|Novartis Investigative Site, Queretaro, 76000, Mexico|Novartis Investigative Site, Groningen, 9713 GZ, Netherlands|Novartis Investigative Site, Nordbyhagen, Oslo, 1478, Norway|Novartis Investigative Site, Bergen, NO-5021, Norway|Novartis Investigative Site, Rostov On Don, 344022, Russian Federation|Novartis Investigative Site, St Petersburg, 197110, Russian Federation|Novartis Investigative Site, Singapore, 169608, Singapore|Novartis Investigative Site, Kosice, 04011, Slovakia|Novartis Investigative Site, Ljubljana, 1000, Slovenia|Novartis Investigative Site, Stockholm, 141 86, Sweden|Novartis Investigative Site, Kaohsiung, 83301, Taiwan|Novartis Investigative Site, New Taipei City, 23561, Taiwan|Novartis Investigative Site, New Taipei, 22060, Taiwan|Novartis Investigative Site, Taichung, 40447, Taiwan|Novartis Investigative Site, Taichung, 407219, Taiwan|Novartis Investigative Site, Taipei, 10002, Taiwan|Novartis Investigative Site, Taoyuan, 33305, Taiwan|Novartis Investigative Site, Bangkok, 10330, Thailand|Novartis Investigative Site, Bangkok, 10400, Thailand|Novartis Investigative Site, Istanbul, TUR, 34098, Turkey|Novartis Investigative Site, Istanbul, 34371, Turkey|Novartis Investigative Site, Kocaeli, 41380, Turkey|Novartis Investigative Site, Mersin, 33110, Turkey|Novartis Investigative Site, Talas Kayseri, 38039, Turkey|Novartis Investigative Site, Cambridge, CB2 0QQ, United Kingdom|Novartis Investigative Site, Leicester, LE5 4PW, United Kingdom|Novartis Investigative Site, London, SE5 9RS, United Kingdom|Novartis Investigative Site, Newcastle upon Tyne, NE7 7DN, United Kingdom|Novartis Investigative Site, Salford, M6 8HD, United Kingdom|Novartis Investigative Site, Ho Chi Minh, VNM, 700000, Vietnam Less <<
NCT06797518 Glomerulonephritis, IGA|Immuno... More >>globulin A Nephropathy Less << PHASE2 NOT_YET_RECRUITING 2028-01-20 -
NCT03896152 Paroxysmal Nocturnal Hemoglobi... More >>nuria Less << PHASE2 COMPLETED 2022-02-09 Novartis Investigative Site, S... More >>eoul, 03080, Korea, Republic of|Novartis Investigative Site, Seoul, 06351, Korea, Republic of|Novartis Investigative Site, Kota Kinabalu, Sabah, 88586, Malaysia|Novartis Investigative Site, Singapore, 119228, Singapore|Novartis Investigative Site, Taipei, 10002, Taiwan Less <<
NCT04747613 Paroxysmal Nocturnal Hemoglobi... More >>nuria Less << PHASE3 ACTIVE_NOT_RECRUITING 2027-10-19 City Of Hope, Duarte, Californ... More >>ia, 91010, United States|USC Norris Cancer Center, Los Angeles, California, 90033, United States|Univ of California Irvine (Chao Family Comprehensive Cancer Center), Orange, California, 92868, United States|Lakes Research, Miami Lakes, Florida, 33014, United States|Augusta University, Augusta, Georgia, 30912, United States|Montefiore Medical Center, Bronx, New York, 10461, United States|Cleveland Clinic Foundation, Cleveland, Ohio, 44195, United States|Prisma Health Upstate, Greenville, South Carolina, 29615, United States|Novartis Investigative Site, Santo Andre, SP, 09090-790, Brazil|Novartis Investigative Site, Sao Paulo, SP, 01323-900, Brazil|Novartis Investigative Site, Beijing, 100730, China|Novartis Investigative Site, Tianjin, 300020, China|Novartis Investigative Site, Tianjin, 300052, China|Novartis Investigative Site, Ostrava, Poruba, 708 52, Czechia|Novartis Investigative Site, Brno Bohunice, 625 00, Czechia|Novartis Investigative Site, Lille, 59037, France|Novartis Investigative Site, Nantes Cedex 1, 44093, France|Novartis Investigative Site, Nice, 06202, France|Novartis Investigative Site, Paris 10, 75475, France|Novartis Investigative Site, Toulouse, 31059, France|Novartis Investigative Site, Aachen, 52074, Germany|Novartis Investigative Site, Dresden, 01307, Germany|Novartis Investigative Site, Essen, 45147, Germany|Novartis Investigative Site, Hamburg, 20246, Germany|Novartis Investigative Site, Riesa, 01589, Germany|Novartis Investigative Site, Ulm, 89081, Germany|Novartis Investigative Site, Ascoli Piceno, AP, 63100, Italy|Novartis Investigative Site, Avellino, AV, 83100, Italy|Novartis Investigative Site, Firenze, FI, 50134, Italy|Novartis Investigative Site, Milano, MI, 20122, Italy|Novartis Investigative Site, Roma, RM, 00161, Italy|Novartis Investigative Site, Torino, TO, 10126, Italy|Novartis Investigative Site, Bassano Del Grappa, Vicenza, 36061, Italy|Novartis Investigative Site, Nagoya, Aichi, 453-8511, Japan|Novartis Investigative Site, Fukushima city, Fukushima, 960 1295, Japan|Novartis Investigative Site, Kanazawa, Ishikawa, 920 8641, Japan|Novartis Investigative Site, Isehara, Kanagawa, 259-1193, Japan|Novartis Investigative Site, Suwa, Nagano, 392-8510, Japan|Novartis Investigative Site, Suita, Osaka, 565 0871, Japan|Novartis Investigative Site, Shinjuku Ku, Tokyo, 160-0023, Japan|Novartis Investigative Site, Kyoto, 606 8507, Japan|Novartis Investigative Site, Niigata, 951 8520, Japan|Novartis Investigative Site, Seoul, 03080, Korea, Republic of|Novartis Investigative Site, Seoul, 06351, Korea, Republic of|Novartis Investigative Site, Vilnius, LT-08661, Lithuania|Novartis Investigative Site, Kota Kinabalu, Sabah, 88586, Malaysia|Novartis Investigative Site, Kuching, Sarawak, 93586, Malaysia|Novartis Investigative Site, Nijmegen, 6500HB, Netherlands|Novartis Investigative Site, Singapore, 119074, Singapore|Novartis Investigative Site, Barcelona, Catalunya, 08036, Spain|Novartis Investigative Site, Santiago De Compostela, Galicia, 15706, Spain|Novartis Investigative Site, San Sebastian, Pais Vasco, 20080, Spain|Novartis Investigative Site, Hualien, 970, Taiwan|Novartis Investigative Site, Taipei, 10002, Taiwan|Novartis Investigative Site, Istanbul, 34093, Turkey|Novartis Investigative Site, Leeds, West Yorkshire, LS9 7TF, United Kingdom|Novartis Investigative Site, London, SE5 9RS, United Kingdom Less <<
NCT04889430 Atypical Hemolytic Uremic Synd... More >>rome Less << PHASE3 RECRUITING 2029-03-29 Uni Of Alabama At Birmingham, ... More >>Birmingham, Alabama, 35233, United States|USC Norris Cancer Center, Los Angeles, California, 90033, United States|Univ of California at Los Angeles, Los Angeles, California, 90095, United States|Univ Cali Irvine ALS Neuromuscular, Orange, California, 92868, United States|Harbor-UCLA Medical Center ., Torrance, California, 90502, United States|Georgetown University Lombardi Cancer Center, Washington, District of Columbia, 20007 2197, United States|University Of Miami, Miami, Florida, 33136, United States|Brigham and Womens Hospital, Boston, Massachusetts, 02115, United States|University of Minnesota, Minneapolis, Minnesota, 55455, United States|WA Uni School Of Med, Saint Louis, Missouri, 63110, United States|Rut Univ for Translational Med Scie, New Brunswick, New Jersey, 08901, United States|University of New Mexico, Albuquerque, New Mexico, 87131-0001, United States|Montefiore Medical Center ., Bronx, New York, 10461, United States|Duke University Medical Center, Durham, North Carolina, 27710, United States|University of Cincinnati, Cincinnati, Ohio, 45267-0585, United States|Cleveland Clinic Foundation, Cleveland, Ohio, 44195, United States|Comprehensive Transplant Ctr at OSU, Columbus, Ohio, 43210, United States|UT Southwestern Medical Center, Dallas, Texas, 75390, United States|Baylor Scott and White Research, Temple, Texas, 76502, United States|Virginia Commonwealth University, Richmond, Virginia, 23298, United States|Novartis Investigative Site, Innsbruck, Tyrol, 6020, Austria|Novartis Investigative Site, Wien, 1090, Austria|Novartis Investigative Site, Fortaleza, CE, 60430 370, Brazil|Novartis Investigative Site, Brasilia, DF, 71635-580, Brazil|Novartis Investigative Site, Belo Horizonte, MG, 30150-221, Brazil|Novartis Investigative Site, Pernambuco, Recife, 50740-900, Brazil|Novartis Investigative Site, Porto Alegre, RS, 90035-074, Brazil|Novartis Investigative Site, Botucatu, SP, 18618-970, Brazil|Novartis Investigative Site, Sao Paulo, SP, 01327 001, Brazil|Novartis Investigative Site, Sao Paulo, SP, 04038-002, Brazil|Novartis Investigative Site, Sao Paulo, SP, 05403 000, Brazil|Novartis Investigative Site, Rio de Janeiro, 22270-60, Brazil|Novartis Investigative Site, Salvador, 40301-155, Brazil|Novartis Investigative Site, Guangzhou, Guangdong, 510080, China|Novartis Investigative Site, Nanjing, Jiangsu, 210009, China|Novartis Investigative Site, Yantai, Shandong, 264000, China|Novartis Investigative Site, Beijing, 100034, China|Novartis Investigative Site, Beijing, 100191, China|Novartis Investigative Site, Beijing, 100730, China|Novartis Investigative Site, Shanghai, 200025, China|Novartis Investigative Site, Shanxi, 710063, China|Novartis Investigative Site, Ostrava, Poruba, 708 52, Czechia|Novartis Investigative Site, Prague 4, 146 24, Czechia|Novartis Investigative Site, Praha, 12808, Czechia|Novartis Investigative Site, Thessaloniki, GR, 570 10, Greece|Novartis Investigative Site, Athens, 115 27, Greece|Novartis Investigative Site, Heraklion Crete, 71110, Greece|Novartis Investigative Site, Hyderabad, Andhra Pradesh, 500012, India|Novartis Investigative Site, Thiruvananthapuram, Kerala, 695011, India|Novartis Investigative Site, Nagpur, Maharashtra, 440015, India|Novartis Investigative Site, Pune, Maharashtra, 411011, India|Novartis Investigative Site, Chandigarh, Punjab, 160012, India|Novartis Investigative Site, Chennai, Tamil Nadu, 600006, India|Novartis Investigative Site, Vellore, Tamil Nadu, 632 004, India|Novartis Investigative Site, Lucknow, Uttar Pradesh, 226014, India|Novartis Investigative Site, Iruma-gun, Saitama, 350-0495, Japan|Novartis Investigative Site, Izumo-city, Shimane, 693 8501, Japan|Novartis Investigative Site, Bunkyo ku, Tokyo, 113 8655, Japan|Novartis Investigative Site, Seoul, 03080, Korea, Republic of|Novartis Investigative Site, Seoul, 03722, Korea, Republic of|Novartis Investigative Site, Seoul, 06591, Korea, Republic of|Novartis Investigative Site, Bratislava, 83305, Slovakia|Novartis Investigative Site, Martin, 03601, Slovakia|Novartis Investigative Site, Ljubljana, 1000, Slovenia|Novartis Investigative Site, Taichung, 40447, Taiwan|Novartis Investigative Site, Taoyuan, 33305, Taiwan|Novartis Investigative Site, London, NW1 2BU, United Kingdom|Novartis Investigative Site, Newcastle upon Tyne, NE7 7DN, United Kingdom Less <<
NCT05086744 Immune Thrombocytopenia (ITP)|... More >>Cold Agglutinin Disease (CAD) Less << PHASE2 TERMINATED 2024-05-17 Massachusetts General Hospital... More >>, Boston, Massachusetts, 02114, United States|Novartis Investigative Site, Essen, 45147, Germany|Novartis Investigative Site, Milano, MI, 20122, Italy|Novartis Investigative Site, Seoul, 06351, Korea, Republic of|Novartis Investigative Site, Barcelona, Catalunya, 08035, Spain|Novartis Investigative Site, Madrid, 28009, Spain|Novartis Investigative Site, Murcia, 30008, Spain|Novartis Investigative Site, London, W12 0HS, United Kingdom Less <<
NCT03832114 Glomerulonephritis PHASE2 COMPLETED 2021-04-23 Novartis Investigative Site, I... More >>owa City, Iowa, 52242, United States|Novartis Investigative Site, Montpellier, 34295, France|Novartis Investigative Site, Paris, 75015, France|Novartis Investigative Site, Essen, 45147, Germany|Novartis Investigative Site, Ranica, BG, 24020, Italy|Novartis Investigative Site, Barcelona, Catalunya, 08035, Spain|Novartis Investigative Site, Madrid, 28041, Spain|Novartis Investigative Site, London, W12 0NN, United Kingdom|Novartis Investigative Site, Newcastle Upon Tyne, NE7 7DN, United Kingdom Less <<
NCT05630001 Paroxysmal Nocturnal Hemoglobi... More >>nuria Less << PHASE3 COMPLETED 2024-10-17 City Of Hope National Med Cent... More >>er, Duarte, California, 91010, United States|USC Norris Cancer Center, Los Angeles, California, 90033, United States|Lakes Research, Miami Lakes, Florida, 33014, United States|Mass Gen Hosp Cancer Center, Boston, Massachusetts, 02114, United States|University Of Minnesota, Minneapolis, Minnesota, 55455, United States|Montefiore Medical Center, Bronx, New York, 10461, United States|Cleveland Clinic Foundation, Cleveland, Ohio, 44195, United States|Prisma Health Upstate, Greenville, South Carolina, 29615, United States|Huntsman Cancer Institute Univ of Utah, Salt Lake City, Utah, 84112 0550, United States|Novartis Investigative Site, Nantes Cedex 1, 44093, France|Novartis Investigative Site, Nice, 06202, France|Novartis Investigative Site, Paris 10, 75475, France|Novartis Investigative Site, Aachen, 52074, Germany|Novartis Investigative Site, Dresden, 01307, Germany|Novartis Investigative Site, Essen, 45147, Germany|Novartis Investigative Site, Ulm, 89081, Germany|Novartis Investigative Site, Firenze, FI, 50134, Italy|Novartis Investigative Site, Bassano Del Grappa, Vicenza, 36061, Italy|Novartis Investigative Site, Seoul, 06351, Korea, Republic of|Novartis Investigative Site, Barcelona, Catalunya, 08036, Spain|Novartis Investigative Site, Istanbul, 34093, Turkey|Novartis Investigative Site, Leeds, West Yorkshire, LS9 7TF, United Kingdom|Novartis Investigative Site, London, SE5 9RS, United Kingdom Less <<
NCT05935215 Atypical Hemolytic Uremic Synd... More >>rome Less << PHASE3 RECRUITING 2029-07-19 Novartis Investigative Site, N... More >>anjing, Jiangsu, 210009, China|Novartis Investigative Site, Beijing, 100034, China|Novartis Investigative Site, Beijing, 100730, China|Novartis Investigative Site, Shanghai, 200025, China|Novartis Investigative Site, Iruma-gun, Saitama, 350-0495, Japan|Novartis Investigative Site, Bunkyo ku, Tokyo, 113 8655, Japan|Novartis Investigative Site, Ankara, 06500, Turkey|Novartis Investigative Site, Izmir, 35340, Turkey|Novartis Investigative Site, Kocaeli, 41380, Turkey|Novartis Investigative Site, Mersin, 33110, Turkey|Novartis Investigative Site, London, NW1 2BU, United Kingdom|Novartis Investigative Site, Newcastle upon Tyne, NE7 7DN, United Kingdom Less <<

Protocol

Bio Calculators
Preparing Stock Solutions 1mg 5mg 10mg

1 mM

5 mM

10 mM

2.37mL

0.47mL

0.24mL

11.83mL

2.37mL

1.18mL

23.67mL

4.73mL

2.37mL

Dissolving Methods
Please choose the appropriate dissolution scheme according to your animal administration guide.For the following dissolution schemes, clear stock solution should be prepared according to in vitro experiments, and then cosolvent should be added in turn:

in order to ensure the reliability of the experimental results, the clarified stock solution can be properly preserved according to the storage conditions; The working fluid for in vivo experiment is recommended to be prepared now and used on the same day;

The percentage shown in front of the following solvent refers to the volume ratio of the solvent in the final solution; If precipitation or precipitation occurs in the preparation process, it can be assisted by heating and/or ultrasound.
Protocol 1
Protocol 2
 

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