HomeAzetidine Derivatives in Drug Design
Azetidines possess a favorable balance between satisfactory stability and strong molecular rigidity, enabling efficient adjustment of pharmacological properties exhibited by molecules containing this moiety. Consequently, azetidine is regarded as a favored framework in the realm of drug discovery.
Drug | Structure | Target | Drug Categories |
Edonerpic maleate | ![]() |
Amyloid-β | Neurotrophic Agents |
Drug | Structure | Target | Drug Categories |
Ezetimibe | ![]() |
LDL-C | Anticholesteremic Agents |
A104063190595-65-498%
(3R,4S)-4-(4-(Benzyloxy)phenyl)-1-(4-fluorophenyl)-3-(3-(4-fluorophenyl)-3-oxopropyl)azetidin-2-oneDrug | Structure | Target | Drug Categories |
Cobimetinib | ![]() |
MEK | Antineoplastic Agents |
Drug | Structure | Target | Drug Categories |
Baricitinib | ![]() |
JAK | Antirheumatic Agents |