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Chemical Structure| 1215721-40-6 Chemical Structure| 1215721-40-6

Structure of CP-809101 HCl
CAS No.: 1215721-40-6

Chemical Structure| 1215721-40-6

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CP-809101 HCl is a potent and selective 5-HT2C receptor agonist with pEC50 of 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors respectively.

Synonyms: CP 809,101 (hydrochloride); CP-809101 hydrochloride

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Product Details of CP-809101 HCl

CAS No. :1215721-40-6
Formula : C15H18Cl2N4O
M.W : 341.24
SMILES Code : ClC1=CC(COC2=NC(N3CCNCC3)=CN=C2)=CC=C1.[H]Cl
Synonyms :
CP 809,101 (hydrochloride); CP-809101 hydrochloride
MDL No. :MFCD10687106

Safety of CP-809101 HCl

GHS Pictogram:
Signal Word:Warning
Hazard Statements:H302-H315-H319-H335
Precautionary Statements:P261-P305+P351+P338

Related Pathways of CP-809101 HCl

GPCR

Isoform Comparison

Biological Activity

Description
CP-809101 is a potent and highly selective agonist for the 5-HT2C receptor, exhibiting pEC50 values of 9.96, 7.19, and 6.81 M for the human 5HT2C, 5HT2B, and 5HT2A receptors, respectively. This compound shows efficacy in inhibiting conditioned avoidance responses in rats and counters the hyperactivity induced by PCP (phencyclidine hydrochloride) and d-amphetamine. Additionally, it demonstrates potential to reduce food and nicotine dependence in rats, making it a valuable agent for antipsychotic and nicotine dependence research[1][2].

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1 mM

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10 mM

2.93mL

0.59mL

0.29mL

14.65mL

2.93mL

1.47mL

29.30mL

5.86mL

2.93mL

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