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Chemical Structure| 170277-31-3 Chemical Structure| 170277-31-3

Structure of Infliximab
CAS No.: 170277-31-3

Chemical Structure| 170277-31-3

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Infliximab is a chimeric IgG1 monoclonal antibody that inhibits TNFα by preventing its binding to receptors. Infliximab has potential for research in rheumatoid arthritis, Crohn's disease, and ulcerative colitis.

Synonyms: Avakine; CT-P13

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Product Details of Infliximab

CAS No. :170277-31-3
M.W : 145.88 kDa
SMILES Code : NONE
Synonyms :
Avakine; CT-P13
MDL No. :N/A

Safety of Infliximab

GHS Pictogram:
Signal Word:Warning
Hazard Statements:H302-H315-H319
Precautionary Statements:P501-P270-P264-P280-P302+P352-P337+P313-P305+P351+P338-P362+P364-P332+P313-P301+P312+P330

Isoform Comparison

Biological Activity

In Vitro:

Cell Line
Concentration Treated Time Description References
CCD18Co cells 10 ng/ml 2 h To assess the impact of OSM on inflammatory responses in intestinal stromal cells, results showed that OSM significantly induced the expression of IL6 and various chemokines PMC5420447
LPMNC from IBD patients 10 µg/mL 18 h To test the effect of Infliximab on the release of inflammatory cytokines in LPMNC from IBD patients, results showed that Infliximab significantly reduced the release of IL-1β, IL-6, TNFα, CCL2, Mip-1α, and IP-10. PMC6145287
NCM460 5 ng/mL 0–60 min To measure the dose-dependent effect of SPINK4 on EGFR phosphorylation PMC11245600
HT-29 5 ng/mL 0–60 min To measure the dose-dependent effect of SPINK4 on EGFR phosphorylation PMC11245600

In Vivo:

Species
Animal Model
Administration Dosage Frequency Description References
Mice C57BL/6J mice Subcutaneous injection 30.75 µg/g Single injection, lasted for 2 weeks To evaluate the causative effect of antibiotic treatment on ADA formation, results showed that mice pretreated with cephalosporins had significantly higher ADA levels compared to those pretreated with macrolides, and germ-free mice produced no detectable ADA. PMC8762017
mice TNBS-induced colitis model intravenous injection 5 mg/kg once daily for 5 days To monitor the effect of anti-tumor necrosis factor α antibody therapy using P-selectin-targeted US imaging, results showed a significant decrease in US signal in treated mice, which correlated well with P-selectin expression levels. PMC3244669
Mice DSS-induced colitis model Intraperitoneal injection 10 mg/kg Single injection, lasting 7 days Infliximab suppressed DSS-induced PUMA expression and colitis, alleviating colonic damage and IEC apoptosis. PMC3083802
Mice TNFdARE mouse model Intraperitoneal injection 100 µg/mouse Twice a week for 15 days To evaluate the efficacy of Infliximab in TNFdARE mice, the results showed that Infliximab significantly suppressed inflammatory gene expression, but histological improvement was not significant. PMC9282884
Mice DSS-induced colitis model Intraperitoneal injection 5 mg/kg 2 consecutive days To evaluate the therapeutic effect of Infliximab on colitis PMC11245600

Clinical Trial:

NCT Number Conditions Phases Recruitment Completion Date Locations
NCT00325078 Chronic Granulomatous Disease|... More >>Crohn'S-like IBD|Inflammatory Bowel Disease (IBD) Less << PHASE1|PHASE2 TERMINATED 2025-06-12 National Institutes of Health ... More >>Clinical Center, 9000 Rockville Pike, Bethesda, Maryland, 20892, United States Less <<
NCT02566889 Inflammatory Bowel Diseases PHASE4 TERMINATED 2025-07-19 Phoenix, Arizona, United State... More >>s|Los Angeles, California, United States|San Francisco, California, United States|Hartford, Connecticut, United States|Wilmington, Delaware, United States|Atlanta, Georgia, United States|Chicago, Illinois, United States|Peoria, Illinois, United States|Indianapolis, Indiana, United States|Shreveport, Louisiana, United States|Portland, Maine, United States|Baltimore, Maryland, United States|Boston, Massachusetts, United States|Waltham, Massachusetts, United States|Rochester, Minnesota, United States|Saint Paul, Minnesota, United States|Kansas City, Missouri, United States|Mineola, New York, United States|New York, New York, United States|Stony Brook, New York, United States|Chapel Hill, North Carolina, United States|Cleveland, Ohio, United States|Philadelphia, Pennsylvania, United States|Pittsburgh, Pennsylvania, United States|Charleston, South Carolina, United States|Dallas, Texas, United States|Fort Worth, Texas, United States|Fairfax, Virginia, United States|Madison, Wisconsin, United States|Vancouver, British Columbia, Canada|Halifax, Nova Scotia, Canada|Hamilton, Ontario, Canada|London, Ontario, Canada|Toronto, Ontario, Canada|Montreal, Quebec, Canada|Sherbrooke, Quebec, Canada Less <<
NCT03192878 Takayasu Arteritis UNKNOWN 2025-07-19 IRCCS Ospedale San Raffaele, M... More >>ilano, MI, 20132, Italy Less <<
NCT00106847 Psoriasis|Parapsoriasis PHASE3 COMPLETED 2025-07-05 -
NCT03765450 Ulcerative Colitis ACTIVE_NOT_RECRUITING 2025-12-24 UCSD, San Diego, California, 9... More >>2037, United States|Cornell University, New York, New York, 10065, United States|London Health Sciences Center, London, Ontario, N6A 5A5, Canada|Mount Sinai Hospital, Toronto, Ontario, M5G 1X5, Canada Less <<
NCT01256489 Stevens-Johnson Syndrome|Corne... More >>al Blindness Less << PHASE1|PHASE2 WITHDRAWN 2025-01-15 Massachusetts Eye and Ear Infi... More >>rmary, Boston, Massachusetts, 02114, United States Less <<
NCT02088944 Serological C Reactive Protein... More >> or Erythrocyte Sedimentation Rate Less << UNKNOWN - -
NCT03937609 Colitis, Ulcerative PHASE4 TERMINATED 2024-12-15 St Vincent's University Hospit... More >>al, Dublin, Ireland|Academic Medical Center, Amsterdam, Netherlands|OLVG Oost, Amsterdam, Netherlands|Radboud UMC, Nijmegen, Netherlands|Klinikk Baerum Sykehus, B?rums Verk, Norway|Akerhus University Hospital, L?renskog, Norway|Helse Stavanger, Stavanger, Norway Less <<
NCT01220518 Ankylosing Spondylitis PHASE1 COMPLETED 2025-06-12 Inha University Hostpital, Inc... More >>heon, Korea, Republic of Less <<
NCT01349920 Crohn Disease COMPLETED 2015-09-28 -
NCT01971814 Ulcerative Colitis (UC)|Inflam... More >>matory Bowel Disease Less << PHASE1 COMPLETED 2025-01-15 University of California at Sa... More >>n Francisco, San Francisco, California, 94143, United States Less <<
NCT06614387 Ulcerative Colitis PHASE3 NOT_YET_RECRUITING 2028-11-30 -
NCT02522169 Pediatric Crohns Disease UNKNOWN 2025-12-16 -
NCT00006292 Rheumatoid Arthritis PHASE2 COMPLETED 2025-09-05 National Institute of Arthriti... More >>s and Musculoskeletal and Skin Diseases (NIAMS), Bethesda, Maryland, 20892, United States Less <<
NCT00201799 Graft-Versus-Host Disease PHASE2 COMPLETED 2025-03-08 Ohio State University, Columbu... More >>s, Ohio, 43210, United States Less <<
NCT05719389 Inflammatory Bowel Diseases|Rh... More >>eumatologic Disease Less << RECRUITING 2025-04-20 Irccs Ospedale San Raffaele, M... More >>ilano, 20132, Italy Less <<
NCT00106834 Psoriasis PHASE3 COMPLETED 2025-10-04 -
NCT02770794 Arthritis, Rheumatoid PHASE4 COMPLETED 2020-08-14 Chiba University Hospital, Chi... More >>ba, 260-8677, Japan Less <<
NCT04312659 Crohn Disease COMPLETED 2023-09-12 Guangzhou Women And Children's... More >> Medical Center, Guangzhou, 510623, China|The Children's Hospital, Zhejiang University School Of Medicine, Hangzhou, 310052, China|Ruijin Hospital, Shanghai Jiao Tong University, Shanghai, 200025, China|Children's Hospital of Fudan University, Shanghai, 201102, China|Henan Children's Hospital, Zhengzhou Children's Hospital, ZhengZhou, 450018, China Less <<
NCT03452501 Inflammatory Bowel Diseases|Cr... More >>ohn Disease|Fistulizing Crohn's Disease|Ulcerative Colitis Less << COMPLETED 2020-08-17 King Abdulaziz University Hosp... More >>ital, Jeddah, Saudi Arabia|Prince Sultan Military Medical City, Riyadh, 11159, Saudi Arabia|King Abdullah International Medical Research Center, Riyadh, 11426, Saudi Arabia|King Saud Medical City, Riyadh, Saudi Arabia Less <<
NCT02505568 Behcet Disease PHASE3 COMPLETED 2018-07-13 Busan, Korea, Republic of|Daeg... More >>u, Korea, Republic of|Gangwon-do, Korea, Republic of|Gyeonggi-do, Korea, Republic of|Seoul, Korea, Republic of Less <<
NCT00236028 Rheumatoid Arthritis PHASE3 COMPLETED 2025-04-03 -
NCT00036439 Ulcerative Colitis PHASE3 COMPLETED 2025-01-07 -
NCT04779892 Rheumatoid Arthritis PHASE1 COMPLETED 2020-06-15 Shanghai Xuhui Central Hospita... More >>l, Shanghai, Shanghai, 200031, China Less <<
NCT00823641 HTLV-I-associated Myelopathy PHASE2 TERMINATED 2025-03-11 Imperial College Healthcare NH... More >>S Trust, London, W2 1PG, United Kingdom Less <<
NCT00462072 Rheumatoid Arthritis|Psoriatic... More >> Arthritis|Psoriasis|Crohn's Disease Less << PHASE4 COMPLETED 2025-08-10 University of Rochester, Roche... More >>ster, New York, 14642, United States Less <<
NCT00741104 Rheumatoid Arthritis COMPLETED 2025-06-08 -
NCT00443222 Refractory Myositis PHASE2|PHASE3 COMPLETED - -
NCT05280405 Inflammatory Bowel Diseases PHASE4 RECRUITING 2025-01-31 Institute for Maternal and Chi... More >>ld Health - IRCCS "Burlo Garofolo", Trieste, 34137, Italy Less <<
NCT00036374 Rheumatoid Arthritis, Juvenile PHASE3 COMPLETED 2025-12-06 -
NCT03445624 Inflammatory Bowel Diseases COMPLETED 2021-10-01 Hyam Fathy, Assiut, Egypt
NCT00033891 Dermatomyositis|Polymyositis PHASE2 COMPLETED 2010-05-20 National Institutes of Health ... More >>Clinical Center, 9000 Rockville Pike, Bethesda, Maryland, 20892, United States Less <<
NCT00076726 Giant Cell Arteritis PHASE2 TERMINATED 2025-07-05 -
NCT01850121 Ankylosing Spondylitis COMPLETED 2025-05-08 Sahlgrenska University Hospita... More >>l, Gothenburg, S-413 45, Sweden Less <<
NCT02799615 Colitis, Ulcerative|Bowel Dise... More >>ases, Inflammatory Less << COMPLETED 2025-11-19 Connecticut Children's Hospita... More >>l Medical Center, Hartford, Connecticut, 06016, United States|Emory University School of Medicine, Atlanta, Georgia, 30322, United States|Cincinnati Children's Hospital Medical Center, Cincinnati, Ohio, 45229, United States|Nationwide Children's Hospital, Columbus, Ohio, 43205, United States|Children's Hospital of Philadelphia, Philadelphia, Pennsylvania, 19104, United States|Rhode Island Hospital, Providence, Rhode Island, 02903, United States|The Hospital for Sick Children, Toronto, Ontario, Canada Less <<
NCT00791557 Pyoderma Gangrenosum|Crohn's D... More >>isease|Ulcerative Colitis|Inflammatory Bowel Disease Less << COMPLETED 2025-02-10 University Hospitals Cleveland... More >> Medical Center, Cleveland, Ohio, 44106, United States Less <<
NCT04272788 Crohn Disease COMPLETED 2019-09-29 SAHWenzhouMU, Wenzhou, Zhejian... More >>g, China Less <<
NCT00523354 Esophagitis PHASE2 COMPLETED 2025-10-07 EE-Clinics, Praxis Roemerhof, ... More >>Olten, SO, 4600, Switzerland Less <<
NCT01661257 Crohn's Disease PHASE3 COMPLETED 2025-06-11 Samsung Medical Center, Seoul,... More >> 135-710, Korea, Republic of Less <<
NCT05340764 Inflammatory Bowel Diseases PHASE4 COMPLETED 2023-05-04 Washington University School o... More >>f Medicine, Saint Louis, Missouri, 63110, United States Less <<
NCT04655729 Crohn Disease UNKNOWN 2023-01-01 MassGeneral for Children, Bost... More >>on, Massachusetts, 02114, United States Less <<
NCT02638701 Aneurysm|Stroke|Vasculitis|Tum... More >>or Necrosis Factor-alpha Less << PHASE1|PHASE2 ENROLLING_BY_INVITATION 2025-12-26 UCSF Medical Center, San Franc... More >>isco, California, 94143, United States Less <<
NCT00571337 Crohn Disease PHASE3 COMPLETED 2025-07-10 Gent University Hospital, Gent... More >>, 9000, Belgium|CHU LIEGE - Sart Tilman, Liege, 4000, Belgium|Chu Amiens, Amiens, 80054, France|Chu Besancon, Besancon, 25030, France|Hopital Saint Andre, Bordeaux, 33075, France|CHU CAEN, Caen, 14033, France|Hopital Beaujon, Clichy, 92110, France|Hopital Louis Mourier, Colombes, 92700, France|Hopital Henri Mondor, Creteil, 94010, France|CHRU Lille, Lille, France|Chu Marseille - Hopital Nord, Marseille, 13915, France|Ch Le Raincy Montfermeil, Montfermeil, 93370, France|Chu Montpellier, Montpellier, 34295, France|Chu Nantes, Nantes, 44093, France|Hopital Lariboisiere, Paris, 75010, France|Hopital Saint Louis, Paris, 75010, France|Hopital Georges Pompidou, Paris, 75015, France|Hopital Haut Leveque, Pessac, 33604, France|CHU LYON, Pierre Benite, 69495, France|Chu Rouen, Rouen, 76031, France|Chu Strasbourg, Strasbourg, 67091, France|Chu Toulouse, Toulouse, 31403, France|Chu Tours, Tours, 37044, France Less <<
NCT05906576 Crohn Disease PHASE4 RECRUITING 2025-02-27 Beijing Children's Hospital, C... More >>apital Medical University, Beijing, China Less <<
NCT02060318 Crohn Disease COMPLETED 2016-03-07 Hvidovre Hospital, Hvidovre, C... More >>openhagen, 2650, Denmark Less <<
NCT01266785 Crohn's Disease WITHDRAWN 2025-07-12 Oregon Health & Science Univer... More >>sity, Portland, Oregon, 97239, United States Less <<
NCT01217086 Rheumatoid Arthritis PHASE3 COMPLETED 2025-07-12 Hanyang University Medical Cen... More >>ter, Seoul, Korea, Republic of Less <<
NCT00075075 Scleritis PHASE1 COMPLETED 2007-09-06 National Institutes of Health ... More >>Clinical Center, 9000 Rockville Pike, Bethesda, Maryland, 20892, United States Less <<
NCT00029042 Juvenile Rheumatoid Arthritis PHASE2 TERMINATED 2025-10-05 National Institute of Arthriti... More >>s and Musculoskeletal and Skin Diseases (NIAMS), Bethesda, Maryland, 20892, United States Less <<
NCT02770040 Ulcerative Colitis PHASE4 COMPLETED 2022-09-07 Austin Health, Melbourne, Vict... More >>oria, 3084, Australia Less <<
NCT04425538 COVID-19 PHASE2 COMPLETED 2021-01-22 Tufts Medical Center, Boston, ... More >>Massachusetts, 02111, United States Less <<
NCT01148901 Ankylosing Spondylitis PHASE4 WITHDRAWN 2025-12-10 -
NCT02605642 Rheumatoid Diseases|Rheumatoid... More >> Arthritis|Ankylosing Spondylitis|Psoriatic Arthritis Less << COMPLETED 2018-12-31 MHAT Trimontium OOD, Plovdiv, ... More >>4000, Bulgaria|MHAT Kaspela EOOD, Plovdiv, 4001, Bulgaria|Diagnostic Consultative Center 17 Sofia EOOD, Sofia, 1233, Bulgaria|Lucere Skin Dermatology & Laser Clinic, Edmonton, Alberta, T6X 0N9, Canada|Nexus Clinical Research, St. John's, Newfoundland and Labrador, A1A 5E8, Canada|Dr. Juris Lazovskis Inc., Sydney, Nova Scotia, B1S 3N1, Canada|The Waterside Clinic, Barrie, Ontario, L4M 6L2, Canada|William Osler Health System, Brampton, Ontario, L6T 3J1, Canada|Adachi Medicine Professional Corporation, Hamilton, Ontario, L8N 1Y2, Canada|K-W Musculoskeletal Research Inc, Kitchener, Ontario, N2M 5N6, Canada|Y. Liu Medicine Professional, Milton, Ontario, L9T 3Z9, Canada|Credit Valley Imaging Associates, Mississauga, Ontario, L5M 2V8, Canada|Oakville Rheumatology & Osteoporosis, Oakville, Ontario, L6M 4J2, Canada|Ottawa Hospital Research Institute, Ottawa, Ontario, K1Y 4G2, Canada|Arthur Karasik Medicine Professional Corporation, Toronto, Ontario, M9C 5N2, Canada|Dr. Sabeen Anwar Medicine Professional Corporation, Windsor, Ontario, N8X 1T3, Canada|Centre Hospitalier de l'Universite de Montreal - Notre-Dame Hospital, Montreal, Quebec, H2L 1S6, Canada|Centre Rhumatologie de l'Est, Rimouski, Quebec, G5L 8W1, Canada|Centre de Recherche Musculo-Squelettique, Trois-Rivières, Quebec, G8Z 1Y2, Canada|Groupe de Recherche en Rhumatologie et Maladies Osseuses (GRMO), Quebec, G1V 3M7, Canada|Revmatolog Mudr. Sirova Klara s.r.o., Ostrava, 701 00, Czechia|Revmatologicky ústav (Rú), Praha 2, 12850, Czechia|Rheumapraxis Steglitz, Berlin, 12163, Germany|Immanuel Diakonie GmbH, Bernau, 16321, Germany|Rheumatologisches MVZ Dresden GmbH, Dresden, 01109, Germany|Asklepios Gesundheitszentrum Elmshorn, Elmshorn, 21073, Germany|Rheumatologische Praxis Dr. med. Kühne, Haldensleben, 39340, Germany|Dr. med. J?rg Kaufmann, Ludwigsfelde, 14974, Germany|Praxis Dr. Herbert Kellner, Muenchen, 80639, Germany|MVZ für Rheumatologie Dr. Martin Welcker GmbH, Planegg, 82152, Germany|Berufsausübungsgemeinschaft Martin Bohl-Bühler & Dr. med. Sabine Reckert, Potsdam, 14469, Germany|Dr. med. Jochen Walter - FA für Innere Medizin Rheumatologe, Rendsburg, 24768, Germany|University General Hospital of Heraklion, Heraklion, Crete, 71110, Greece|Complexo Hospitalario Universitario A Coru?a, A Coru?a A Coru?a, 15006, Spain|Hospital Universitario Vall d'Hebron, Barcelona, 08035, Spain|Hospital Universitario de Canarias, San Cristóbal de La Laguna, 38320, Spain|Portsmouth Hospitals NHS Trust - Queen Alexandra Hospital, Portsmouth, PO6 3LY, United Kingdom|Salisbury NHS Foundation Trust - Salisbury District Hospital, Sailsbury, SP2 8BJ, United Kingdom Less <<
NCT00051623 Arthritis, Psoriatic PHASE3 COMPLETED 2025-06-04 -
NCT00056264 Chronic Obstructive Pulmonary ... More >>Disease|COPD Less << PHASE3 COMPLETED 2025-12-04 -
NCT00724243 Rheumatoid Arthritis COMPLETED 2025-10-08 -
NCT05552287 Crohn Disease|Child, Only|Biol... More >>ogic; Inadequate Less << PHASE4 RECRUITING 2025-08-25 Erasmus Medical Center, Rotter... More >>dam, 3015 GD, Netherlands Less <<
NCT06274294 Inflammatory Bowel Diseases PHASE3 RECRUITING 2025-01-25 Institut des MICI, Neuilly-sur... More >>-Seine, 92200, France Less <<
NCT03209232 Ulcerative Colitis TERMINATED 2021-09-01 Schenider Children's Medical C... More >>enter, Peta? Tiqwa, 4920235, Israel Less <<
NCT00096655 Ulcerative Colitis PHASE3 COMPLETED 2025-08-07 -
NCT00073437 Sarcoidosis PHASE3 COMPLETED 2025-02-05 -
NCT00228839 Graft vs Host Disease PHASE1 COMPLETED 2025-10-06 Children's Healthcare of Atlan... More >>ta/Emory University, Atlanta, Georgia, 30322, United States Less <<
NCT04835506 Crohn Disease|Ulcerative Colit... More >>is|Inflammatory Bowel Diseases Less << PHASE4 ENROLLING_BY_INVITATION 2024-12-31 Yale University School of Medi... More >>cine, New Haven, Connecticut, 06510, United States|University of Miami, Miami, Florida, 33136, United States|University of Chicago Medicine, Chicago, Illinois, 60637, United States|Northwestern University, Evanston, Illinois, 60208, United States|Rockford GI, Rockford, Illinois, 61107, United States|University of Maryland Medical Center, Baltimore, Maryland, 21201, United States|Boston Children's Hospital, Boston, Massachusetts, 02115, United States|Beth Israel Deaconess Medical Center, Boston, Massachusetts, 02215, United States|Lahey Hospital and Medical Center, Burlington, Massachusetts, 01805, United States|University of Minnesota, Minneapolis, Minnesota, 55455, United States|Dartmouth-Hitchcock Medical Center, Lebanon, New Hampshire, 03766, United States|NYU Langone Health, New York, New York, 10016, United States|Icahn School of Medicine at Mount Sinai, New York, New York, 10029, United States|Weill Cornell Medical College, New York, New York, 10065, United States|Atrium Health Center for Digestive Health, Charlotte, North Carolina, 28204, United States|Cleveland Clinic, Cleveland, Ohio, 44195, United States|Children's Hospital of Philadelphia, Philadelphia, Pennsylvania, 19104, United States|LifeSpan Brown University, Providence, Rhode Island, 02915, United States|Medical University of South Carolina, Charleston, South Carolina, 29425, United States|Vanderbilt University Medical Center, Nashville, Tennessee, 20500, United States|University of Texas Southwestern Medical Center, Dallas, Texas, 75390, United States|University of Utah, Salt Lake City, Utah, 84132, United States|Medical College of Wisconsin, Milwaukee, Wisconsin, 53226, United States|London Health Sciences Centre - Children's Hospital, London, Canada|McGill University Health Centre (MUHC) Montreal General Hospital, Montreal, Canada Less <<
NCT00036387 Arthritis, Rheumatoid PHASE3 COMPLETED 2025-11-03 -
NCT01408810 Ulcerative Colitis PHASE4 COMPLETED 2025-11-12 Hospital de S?o Jo?o, Porto, 4... More >>200-319, Portugal Less <<
 

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