Home Cart Sign in  
Chemical Structure| 1661854-97-2 Chemical Structure| 1661854-97-2

Structure of Zipalertinib
CAS No.: 1661854-97-2

Chemical Structure| 1661854-97-2

*Storage: {[sel_prStorage]}

*Shipping: {[sel_prShipping]}

,{[proInfo.pro_purity]}

Zipalertinib is a novel EGFR mutation inhibitor specifically targeting certain EGFR mutations present in tumors. It has significant potential in treating various EGFR mutation-related cancers, such as non-small cell lung cancer.

Synonyms: TAS6417; CLN-081

4.5 *For Research Use Only !

{[proInfo.pro_purity]}
Cat. No.: {[proInfo.prAm]} Purity: {[proInfo.pro_purity]}

Change View

Size Price VIP Price

US Stock

Global Stock

In Stock
{[ item.pr_size ]} Inquiry {[ getRatePrice(item.pr_usd,item.pr_rate,item.mem_rate,item.pr_is_large_size_no_price, item.vip_usd) ]}

US Stock: ship in 0-1 business day
Global Stock: ship in 5-7 days

  • {[ item.pr_size ]}

In Stock

- +

Please Login or Create an Account to: See VIP prices and availability

US Stock: ship in 0-1 business day
Global Stock: ship in 2 weeks

  • 1-2 Day Shipping
  • High Quality
  • Technical Support
Product Citations

Alternative Products

Product Details of Zipalertinib

CAS No. :1661854-97-2
Formula : C23H20N6O
M.W : 396.44
SMILES Code : C=CC(N[C@@H]1CN2C3=NC=NC(N)=C3C(C4=CC5=CC=CC=C5N=C4)=C2C(C)=C1)=O
Synonyms :
TAS6417; CLN-081
MDL No. :MFCD31715430
InChI Key :MKCYPWYURWOKST-INIZCTEOSA-N
Pubchem ID :117918742

Safety of Zipalertinib

GHS Pictogram:
Signal Word:Warning
Hazard Statements:H302-H315-H319-H335
Precautionary Statements:P261-P280-P301+P312-P302+P352-P305+P351+P338

Related Pathways of Zipalertinib

RTK
JAK-STAT

Isoform Comparison

Biological Activity

Target
  • EGFR/ErbB1

    EGFR (L861Q), IC50:4.1 nM

    EGFR WT, IC50:8 nM

  • ErbB4

    HER4, IC50:4 nM

  • mutant EGFR

    EGFR L858R, IC50:2 nM

    EGFR(d746-750), IC50:1.4 nM

In Vitro:

Cell Line
Concentration Treated Time Description References
BEAS-2B 10 μM 72 h Evaluate the toxicity of TAS6417 on normal cells, results showed that 10 μM TAS6417 and erlotinib had no impact on BEAS-2B cells PMC6872223

In Vivo:

Species
Animal Model
Administration Dosage Frequency Description References
BALB/cAJcl-nu/nu mice Subcutaneous implantation model Oral 50, 100, 200 mg/kg Once daily for 10-14 days Evaluate the inhibitory effect of TAS6417 on EGFR mutations in vivo, results showed that TAS6417 at doses of 50, 100, 200 mg/kg/day significantly inhibited tumor growth PMC6872223

Clinical Trial:

NCT Number Conditions Phases Recruitment Completion Date Locations
NCT05967689 Advanced or Metastatic NSCLC H... More >>arboring Epidermal Growth Factor Receptor (EGFR) Exon 20 Insertion (ex20ins) Mutations Less << PHASE2 ACTIVE_NOT_RECRUITING 2025-10-20 O'Neal Comprehensive Cancer Ce... More >>nter at the University of Alabama at Birmingham, Birmingham, Alabama, 35294, United States|City of Hope - Duarte (Main Campus), Duarte, California, 91010, United States|City of Hope - Huntington Beach, Huntington Beach, California, 92648, United States|City of Hope Orange County Lennar Foundation Cancer Center, Irvine, California, 92618, United States|SCRI - Florida Cancer Specialists - East Region Research Office, West Palm Beach, Florida, 33401, United States|Beth Israel Deaconess Medical Center, Boston, Massachusetts, 02115, United States|Comprehensive Cancer Centers of Nevada - Henderson, Henderson, Nevada, 89052, United States|Comprehensive Cancer Centers of Nevada - Horizon Ridge Henderson, Henderson, Nevada, 89052, United States|Comprehensive Cancer Centers of Nevada - Southeast Henderson - Stephanie, Henderson, Nevada, 89074, United States|Comprehensive Cancer Centers of Nevada - Northwest, Las Vegas, Nevada, 89128, United States|Comprehensive Cancer Centers of Nevada - Summerlin Medical Center II, Las Vegas, Nevada, 89144, United States|Comprehensive Cancer Centers of Nevada - Southwest, Las Vegas, Nevada, 89148, United States|Comprehensive Cancer Centers of Nevada - Central Valley - Twain, Las Vegas, Nevada, 89169, United States|Memorial Sloan Kettering Cancer Center - Basking Ridge, Basking Ridge, New Jersey, 07920, United States|Memorial Sloan Kettering Cancer Center - Monmouth, Middletown, New Jersey, 07748, United States|Memorial Sloan Kettering Cancer Center - Bergen, Montvale, New Jersey, 07645, United States|Memorial Sloan Kettering Cancer Center - Commack, Commack, New York, 11725, United States|Memorial Sloan Kettering Cancer Center - Westchester, Harrison, New York, 10604, United States|Memorial Sloan Kettering Cancer Center - New York, New York, New York, 10065, United States|Memorial Sloan Kettering Cancer Center - Nassau, Uniondale, New York, 11553, United States|Gabrail Cancer and Research Center, Canton, Ohio, 44718, United States|SCRI - Mark H. Zangmeister Cancer Center, Columbus, Ohio, 43219, United States|The Toledo Clinic Cancer Center, Toledo, Ohio, 43623, United States|Tennessee Oncology - Nashville - Centennial Clinic - Medical Oncology, Nashville, Tennessee, 37203, United States|University of Texas MD Anderson Cancer Center, Houston, Texas, 77030, United States|Virginia Cancer Specialists - Arlington Office, Arlington, Virginia, 22205, United States|Virginia Cancer Specialists - Fairfax Office, Fairfax, Virginia, 22031, United States|Virginia Cancer Specialists - Gainesville Office, Gainesville, Virginia, 20155, United States|Virginia Cancer Specialists - Reston, Reston, Virginia, 20190, United States|Froedtert and Medical College of Wisconsin, Milwaukee, Wisconsin, 53226, United States|Bankstown-Lidcombe Hospital, Bankstown, New South Wales, 2200, Australia|GenesisCare - North Shore, Saint Leonards, New South Wales, 2065, Australia|Joondalup Health Campus, Joondalup, Western Australia, 6027, Australia|William Osler Health System - Brampton Civic Hospital, Brampton, L6R 3J7, Canada|Les H?pitaux Universitaires de Strasbourg, Strasbourg cedex, Aslace, 67091, France|H?pital C?te De Nacre, Caen cedex 9, Basse-Normandie, 14033, France|Institut Curie, Paris cedex 05, Ile-de-France, 75248, France|Centre Hospitalier Universitaire Limoges, Limoges cedex, Limousin, 87042, France|Centre Hospitalier Universitaire De Nantes - H?pital Nord Laennec, Saint-Herblain, Loire-Atlantique, 44805, France|H?pital Haut-Lévêque, Pessac, Nouvelle-Aquitaine, 33604, France|H?pital Nord de Marseille, Marseille, Provence Alpes Cote d′Azur, 13015, France|Centre Léon Bérard, Lyon, Rhone-Alpes, 69008, France|H?pital Ambroise-Paré, Boulogne-Billancourt, ?le-de-France, 92100, France|Klinikum Kassel, Kassel, Hassen, 34125, Germany|Universit?tsklinikum Gie?en und Marburg - Gie?en, Gie?en, Hessen, 35392, Germany|Universitatsklinikum Carl Gustav Carus Dresden, Dresden, SAchsen, 01301, Germany|Universit?tsklinikum Regensburg, Regensburg, 93053, Germany|Queen Mary Hospital - Hong Kong, Pok Fu Lam, Hong Kong Island, Hong Kong|Azienda Ospedaliero - Universitaria Careggi, Firenze, Florence, 50134, Italy|Istituto Romagnolo per lo Studio dei Tumori "Dino Amadori" - IRST, Meldola, Forli-Cesena, 47014, Italy|Azienda Socio-Sanitaria Territoriale di Cremona, Cremona, 26100, Italy|Istituto di Ricovero e Cura a Carattere Scientifico (IRCCS) - Ospedale San Raffaele, Milan, 20132, Italy|Azienda Ospedaliero-Universitaria di Parma, Parma, 43126, Italy|Azienda Unità Sanitaria Locale della Romagna, Ravenna, 48121, Italy|Aichi Cancer Center, Nagoya, Aiti, 464-8681, Japan|Kyushu Cancer Center, Fukuoka-shi, Hukuoka, 811-1395, Japan|Sendai Kousei Hospital, Sendai, Miyagi, 980-0873, Japan|Kindai University Hospital, ōsaka-sayama-Shi, Osaka, 589-8511, Japan|Shizuoka Cancer Center, Sunto-gun, Sizuoka, 411-8777, Japan|National Cancer Center Hospital East, Kashiwa-shi, Tiba, 277-8577, Japan|Cancer Institute Hospital of JFCR, Koto, Tokyo, 135-8550, Japan|Niigata Cancer Center Hospital, Niigata, 951-8566, Japan|Okayama University Hospital, Okayama, 700-8558, Japan|National Cancer Center Hospital, Tokyo, 104-0045, Japan|Seoul National University Bundang Hospital, Seongnam-si, Gyeonggi-Do, 13620, Korea, Republic of|Catholic University of Korea Saint Vincent's Hospital, Suwon-si, Gyeonggi-do, 16247, Korea, Republic of|Ajou University Hospital, Suwon-si, Gyeonggi-do, 16499, Korea, Republic of|Gyeongsang National University Hospital, Jinju, Gyeongsangnamdo [Kyongsangnam-do], 52727, Korea, Republic of|Inha University Hospital, Incheon, Incheon Gwang'yeogsi [Inch'on-Kwangyokshi], 22332, Korea, Republic of|Chonnam National University Hwasun Hospital, Hwasun, Jeollanam-do, 58128, Korea, Republic of|Asan Medical Center, Seoul, Seoul Teugbyeolsi [Seoul-T'ukpyolshi], 05505, Korea, Republic of|Korea University Guro Hospital, Seoul, Seoul Teugbyeolsi [Seoul-T'ukpyolshi], 08308, Korea, Republic of|The Catholic University of Korea - Seoul St. Mary's Hospital, Soeul, Seoul Teugbyeolsi [Seoul-T'ukpyolshi], 06591, Korea, Republic of|Hospital Regional Universitario de Málaga - Hospital General, Málaga, Malaga, 29010, Spain|Clínica Mi Tres Torres, Barcelona, 08017, Spain|Hospital Quirónsalud Barcelona, Barcelona, 08023, Spain|Hospital Universitario de Jaén, Jaén, 23007, Spain|MD Anderson Cancer Center Madrid, Madrid, 28033, Spain|Hospital Universitario Fundación Jiménez Díaz, Madrid, 28040, Spain|Hospital Universitario 12 de Octubre, Madrid, 28041, Spain|Hospital Universitario La Paz, Madrid, 28046, Spain|T.C. Saglik Bakanligi Ankara Bilkent Sehi?r Hastanesi?, Cankaya, Ankara, 06800, Turkey|Ankara Il Saglik Mudurlugu SBU Gulhane Egitim Ve Arastirma Hastanesi, Etlik, Ankara, 06010, Turkey|Istinye üniversite Hastanesi Liv Hospital Bahcesehir, Esenyurt, Istanbul, 34517, Turkey|Trakya üniversitesi Saglik Arastirma ve Uygulama Merkezi, Edirne, 22030, Turkey|Bagcilar Medipol Mega Universite Hastanesi, Istanbul, 34214, Turkey|T.C. Saglik Bakanligi - Istanbul Il Saglik Mudurlugu - Goztepe Prof. Dr. Suleyman Yalcin Sehir Hastanesi, Istanbul, 34722, Turkey|The Christie NHS Foundation Trust, Manchester, England, M20 4BX, United Kingdom|Nottingham University Hospitals NHS Trust, Nottingham, England, NG5 1PB, United Kingdom Less <<
NCT05973773 Advanced or Metastatic NSCLS W... More >>ith Exon 20 Insertion Mutation Less << PHASE3 RECRUITING 2026-08-24 Comprehensive Cancer Centers o... More >>f Nevada - Henderson, Henderson, Nevada, 89052, United States|Comprehensive Cancer Centers of Nevada - Horizon Ridge Henderson, Henderson, Nevada, 89052, United States|Comprehensive Cancer Centers of Nevada - Southeast Henderson - Stephanie, Henderson, Nevada, 89074, United States|Comprehensive Cancer Centers of Nevada - Summerlin Medical Center II, Las Vegas, Nevada, 89144, United States|Comprehensive Cancer Centers of Nevada - Southwest, Las Vegas, Nevada, 89148, United States|Comprehensive Cancer Centers of Nevada - Central Valley - Twain, Las Vegas, Nevada, 89169, United States|Comprehensive Cancer Centers of Nevada - Northwest, Las Vegas, Nevada, 89218, United States|Gabrail Cancer and Research Center, Canton, Ohio, 44718, United States|The Toledo Clinic Cancer Center, Toledo, Ohio, 43623, United States|University of Texas MD Anderson Cancer Center, Houston, Texas, 77030, United States|Universitair Ziekenhuis Leuven - Campus Gasthuisberg, Leuven, Flemish Brabant, 3000, Belgium|Algemeen Ziekenhuis Maria Middelares, Gent, Oost-Vlaaderen, 9000, Belgium|Algemeen Ziekenhuis Delta - Campus Menen, Menen, West Flanders, 8930, Belgium|Algemeen Ziekenhuis Delta - Campus Rumbeke, Rosières, West-Vlaanderen, 8800, Belgium|Centro Regional Integrado de Oncologia, Fortaleza, Ceará, 60335-480, Brazil|Hospital S?o Lucas da PUCRS, Porto Alegre, Rio Grande Do Sul, 90610-000, Brazil|Clínica Neoplasias Litoral, Itajaí, Santa Catatina, 88301, Brazil|Hospital Amaral Carvalho, Jaú, S?o Paulo, 17210-180, Brazil|Multi-profile Hospital for Active Treatment Uni Hospital, Panagyurishte, Pazardzhik, 1527, Bulgaria|University Multiprofile Hospital for Active Treatment Tsaritsa Yoanna-ISUL, Sofia, 4500, Bulgaria|William Osler Health System - Brampton Civic Hospital, Brampton, Ontario, L6R 3J7, Canada|Princess Margaret Cancer Centre, Toronto, Ontario, M5G 2M9, Canada|Les H?pitaux Universitaires de Strasbourg, Strasbourg cedex, Alsace, 67091, France|H?pital C?te De Nacre, Caen cedex 9, Basse-Normandie, 14033, France|Institut Curie, Paris cedex, Ile-de-France, 75248, France|Centre Hospitalier Universitaire Limoges, Limoges, Limousin, 87042, France|H?pital Haut-Lévêque, Pessac, Nouvelle-Aquitaine, 33604, France|Centre Hospitalier Le Mans, Le Mans cedex 9, Pays De La Loire, 72037, France|H?pital Ambroise-Paré, Boulogne-Billancourt, ?le-de-France, 92100, France|Asklepios Klinik Altona, Hamburg, Hamburg (Hansestadt), 22763, Germany|Universit?tsklinikum Gie?en und Marburg - Gie?en, Gie?en, Hessen, 35392, Germany|LMU Klinikum - Campus Innenstadt, München, 80337, Germany|Universit?tsklinikum Regensburg, Regensburg, 93053, Germany|General Hospital for Thoracic Diseases Sotiria, Athens, Attica, 11527, Greece|Metropolitan General, Piraeus, Attica, 18547, Greece|University General Hospital of Patras, Patra, Peloponnese, 26504, Greece|Metropolitan Hospital, Peiraias, Pireas, 185 47, Greece|University General Hospital of Larissa, Larissa, Thessaly, 41110, Greece|BioClinic Thessaloniki, Thessaloniki, 54622, Greece|Emek Medical Center, Afula, 18101, Israel|Shaare Zedek Medical Center, Jerusalem, 9103102, Israel|Hadassah University Hospital Ein Kerem, Jerusalem, 9112001, Israel|Tel Aviv Sourasky Medical Center, Tel Aviv, 6423906, Israel|Assuta Hospital - Ramat HaHayal, Tel aviv, 69710, Israel|Istituto Romagnolo per lo Studio dei Tumori "Dino Amadori" - IRST, Meldola, Forlì-Cesena, 47014, Italy|Istituto di Ricovero e Cura a Carattere Scientifico (IRCCS) - Ospedale San Raffaele, Milan, 20132, Italy|Azienda Ospedaliero - Universitaria di Modena, Modena, 41224, Italy|Fondazione IRCCS Policlinico San Matteo, Pavia, 27100, Italy|Azienda Unità Sanitaria Locale della Romagna, Ravenna, 48121, Italy|Azienda Ospedaliera Universitaria Integrata Verona, Verona, 37126, Italy|Aichi Cancer Center, Nagoya, Aiti [Aichi], 464-8681, Japan|Hirosaki University Hospital, Hirosaki-Shi, Aomori, 036-8563, Japan|Kyushu Cancer Center, Fukuoka-shi, Hukuoka, 811-1395, Japan|Kitasato University Hospital, Sagamihara, Kanagawa, 252-0375, Japan|Kanagawa Cardiovascular and Respiratory Center, Yokohama, Kanagawa, 236-0051, Japan|Saiseikai Kumamoto Hospital, Kumamoto-Shi, Kumamoto, 861-4163, Japan|Sendai Kousei Hospital, Sendai, Miyagi, 980-0873, Japan|Okayama University Hospital, Okayamashi, Okayama, 700-8558, Japan|Kansai Medical University Hospital, Hirakata, Osaka, 573-1191, Japan|National Hospital Organization Kinki-Chuo Chest Medical Center, Sakai-Shi, Osaka, 591-8555, Japan|Cancer Institute Hospital of JFCR, Koto, Tokyo, 135-8550, Japan|Keio University Hospital, Shinjuku-Ku, Tokyo, 160-8582, Japan|Kanazawa University Hospital, Kanazawa, 920-8641, Japan|Osaka City General Hospital, Osaka, 534-0021, Japan|Osaka Prefectural Hospital Organization - Osaka International Cancer Institute, Osaka, 541-8567, Japan|Catholic University of Korea Saint Vincent's Hospital, Suwon-si, Gyeonggi-do, 16247, Korea, Republic of|Ajou University Hospital, Suwon-si, Gyeonggi-do, 16499, Korea, Republic of|Gyeongsang National University Hospital, Jinju, Gyeongsangnamdo [Kyongsangnam-do], 52727, Korea, Republic of|Inha University Hospital, Incheon, Incheon Gwang'yeogsi [Inch'on-Kwangyokshi], 22332, Korea, Republic of|Korea University Anam Hospital, Seoul, Seoul Teugbyeolsi [Seoul-T'ukpyolshi], 02841, Korea, Republic of|Korea University Guro Hospital, Seoul, Seoul Teugbyeolsi [Seoul-T'ukpyolshi], 08308, Korea, Republic of|Radboud Universitair Medisch Centrum, Nijmegen, Gelderland, 6525 GA, Netherlands|Vrije Universiteit Medisch Centrum, Amsterdam, Noord-Holland, 1081 HV, Netherlands|St. Luke's Medical Center - Quezon City, Quezon City, Metropolitan Manila, 1112, Philippines|Samodzielny Publiczny Szpital Kliniczny Nr 4 w Lublinie, Lublin, Lubelskie, 20-954, Poland|Instytut MSF, ?ód?, Lódzkie, 90-302, Poland|Wielkopolskie Centrum Pulmonologii i Torakochirurgii im. Eugenii i Janusza Zeylandów, Pozna?, Wielkopolskie, 60-569, Poland|Tan Tock Seng Hospital, Singapore, 30433, Singapore|Complejo Hospitalario Universitario A Coru?a, A Coru?a, La Coru?a, 15006, Spain|Clínica Mi Tres Torres, Barcelona, 08017, Spain|Hospital Quirónsalud Barcelona, Barcelona, 08023, Spain|Hospital Clinic de Barcelona, Barcelona, 08036, Spain|Hospital Universitario de Jaén, Jaén, 23007, Spain|MD Anderson Cancer Center Madrid, Madrid, 28033, Spain|Hospital Universitario Fundación Jiménez Díaz, Madrid, 28040, Spain|Hospital Universitario 12 de Octubre, Madrid, 28041, Spain|Hospital Universitario La Paz, Madrid, 28046, Spain|Hospital Regional Universitario de Málaga - Hospital General, Málaga, 29010, Spain|Faculty of Medicine Siriraj Hospital, Bang Phlat, Bangkok, 10700, Thailand|King Chulalongkorn Memorial Hospital, Pathum Wan, Bangkok, 10330, Thailand|Navamindradhiraj University - Faculty of Medicine Vajira Hospital, Krung Thep Maha Nakhon, Khet Dusit, 10300, Thailand|T.C. Saglik Bakanligi Adana Sehir Egitim ve Arastirma Hastanesi, Adana, 01060, Turkey|Medical Park Seyhan Hastanesi, Adana, 01120, Turkey|Hacettepe üniversitesi Kanser Enstitüsü, Ankara, 06010, Turkey|Memorial Ankara Hastanesi, Ankara, 6520, Turkey|Trakya üniversitesi Sa?l?k Ara?t?rma ve Uygulama Merkezi, Edirne, 22130, Turkey|Ankara Il Saglik Mudurlugu SBU Gulhane Egitim Ve Arastirma Hastanesi, Etlik, 06010, Turkey|Bagcilar Medipol Mega Universite Hastanesi, Istanbul, 34214, Turkey|T.C. Saglik Bakanligi - Istanbul Il Saglik Mudurlugu - Goztepe Prof. Dr. Suleyman Yalcin Sehir Hastanesi, Istanbul, 34722, Turkey|T.C. Saglik Bakanligi Ankara Bilkent Sehi?r Hastanesi?, ?ankaya, 06800, Turkey|Royal Free London NHS Foundation Trust, London, England, NW3 2QG, United Kingdom|Nottingham University Hospitals NHS Trust, Nottingham, England, NG5 1PB, United Kingdom|Torbay and South Devon NHS Foundation Trust, Torquay, England, TQ2 7AA, United Kingdom Less <<
NCT04036682 Non Small Cell Lung Cancer|EGF... More >>R Exon 20 Mutation Less << PHASE1|PHASE2 ACTIVE_NOT_RECRUITING 2025-12-24 Pacific Cancer Medical Center,... More >> Inc, Anaheim, California, 92801, United States|City of Hope Comprehensive Cancer Center, Duarte, California, 91010, United States|City of Hope at Irvine Lennar, Irvine, California, 92618, United States|Pacific Shores Medical Group, Long Beach, California, 90813, United States|AdventHealth, Orlando, Florida, 32804, United States|Massachusetts General Hospital, Boston, Massachusetts, 02114, United States|University of Michigan Health System - University Hospital, Ann Arbor, Michigan, 48109, United States|Summit Medical Group PA, Florham Park, New Jersey, 07932, United States|Perlmutter Cancer Center at NYU Langone Hospital - Long Island, Mineola, New York, 11501, United States|New York University Langone Health, New York, New York, 10016, United States|Columbia University Irving Medical Center, New York, New York, 10032, United States|Memorial Sloan Kettering Cancer Center, New York, New York, 10065, United States|Gabrail Cancer Center Research, Canton, Ohio, 44701, United States|Providence Cancer Center, Portland, Oregon, 97213, United States|Providence Oncology & Hematology Care Clinic-Westside, Portland, Oregon, 97225, United States|UPMC Hillman Cancer Center, Pittsburg, Pennsylvania, 15232, United States|Medical University of South Carolina, Charleston, South Carolina, 29425, United States|Virginia Cancer Specialists, Fairfax, Virginia, 22031, United States|Hong Kong University - Queen Mary Hospital, Hong Kong, Hong Kong|Azienda Ospedaliero Universitaria Careggi, Careggi, Italy|Azienda Ospedaliero Universitaria Ospedali Riuniti Umberto I, Marche, Italy|Istituto Scientifico Romagnolo per lo Studio e la Cura dei Tumori (IRST) IRCCS, Meldola, Italy|IRCCS-Istituto Europeo di Oncologia, Milano, Italy|Azienda Ospedaliero Universitaria Modena, Modena, Italy|San Gerardo Hospital, Monza, Italy|Ospedale Santa Maria delle Croci, Ravenna, Italy|National Cancer Center Hospital East, Chiba, Japan|Niigata Cancer Center, Niigata, Japan|Osaka City General Hospital, Osaka, Japan|Osaka International Cancer Institute, Osaka, Japan|Shizuoka Cancer Center, Shizuoka, Japan|National Cancer Center Hospital, Tokyo, Japan|The Cancer Institute Hospital of Japanese Foundation for Cancer Research, Tokyo, Japan|National Cancer Center, Goyang-si, Korea, Republic of|Seoul National University Bundang Hospital (SNUBH), Gyeonggi-do, Korea, Republic of|Gachon University Gil Medical Center, Incheon, Korea, Republic of|Inha University Hospital, Incheon, Korea, Republic of|Samsung Medical Center, Seoul, Korea, Republic of|Asan Medical Center (AMC), Soeul, Korea, Republic of|Korea University Guro Hospital, Soeul, Korea, Republic of|Ajou University Hospital, Suwon-si, Korea, Republic of|The Catholic University Of Korea St. Vincent's Hospital, Suwon-si, Korea, Republic of|The Netherlands Cancer Institute (NKI), Amsterdam, 1066 CX, Netherlands|Leiden University Medical Center, Leiden, 2333 ZA, Netherlands|Singapore Clinical Research Institute, Singapore, 138669, Singapore|National Cancer Centre Singapore, Singapore, 169610, Singapore|University Hospital A Coruna, A Coru?a, Spain|Hospital Clinic i Provincial de Barcelona, Barcelona, Spain|Hospital Parc Tauli, Barcelona, Spain|Hospital Universitario Vall d'Hebron, Barcelona, Spain|Institut Catala d'Oncologia l'Hospitalet, Barcelona, Spain|START Barcelona, Barcelona, Spain|Complejo Hospitalario Universitario Insular Materno Infantil, Las Palmas, Spain|Hospital General Universitario Gregorio Maranon (HGUGM), Madrid, Spain|Hospital Universitario Puerta de Hierro de Majadahonda, Madrid, Spain|University Hospital Quironsalud Madrid, Madrid, Spain|Hospital Regional Universitario de Malaga, Málaga, Spain|Clinica Universidad de Navarra, Pamplona, Spain|Universitat de Valencia - Hospital Universitari i Politecnic La Fe de Valencia (Hospital La Fe Bulevar Sur), Valencia, Spain|Chang Gung Medical Foundation Chiayi Chang Gung Memorial Hospital, Chiayi City, Taiwan|Chung Shan Medical University Hospital, Taichung, Taiwan|Taichung Veterans General Hospital, Taichung, Taiwan|National Taiwan University Hospital, Taipei, 10002, Taiwan|Taipei Medical University Hospital, Taipei, Taiwan Less <<

Protocol

Bio Calculators
Preparing Stock Solutions 1mg 5mg 10mg

1 mM

5 mM

10 mM

2.52mL

0.50mL

0.25mL

12.61mL

2.52mL

1.26mL

25.22mL

5.04mL

2.52mL

Dissolving Methods
Please choose the appropriate dissolution scheme according to your animal administration guide.For the following dissolution schemes, clear stock solution should be prepared according to in vitro experiments, and then cosolvent should be added in turn:

in order to ensure the reliability of the experimental results, the clarified stock solution can be properly preserved according to the storage conditions; The working fluid for in vivo experiment is recommended to be prepared now and used on the same day;

The percentage shown in front of the following solvent refers to the volume ratio of the solvent in the final solution; If precipitation or precipitation occurs in the preparation process, it can be assisted by heating and/or ultrasound.
Protocol 1
Protocol 2

References

 

Historical Records

Categories